SCHEMBL31190888

SCHEMBL31190888

COC(=O)c1ccn2c(Br)c(-c3ccccc3-c3ccc(C)cc3C)nc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.42
AKT2 P31751 2/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPK10 P53779 1/20 0.40
TP53 P04637 2/20 0.38
MAPT P10636 4/20 0.38
GAA P10253 3/20 0.38
ALPL P05186 1/20 0.38
CGAS Q8N884 1/20 0.38
PLAU P00749 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31190932 0.81 ALDH1A1 (0.38) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL31190943 0.77 RAB9A (0.45) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL31091925 0.76 AKT1 (0.46) AKT1AKT2NPC1RAB9ASMN1; SMN2
SCHEMBL31190916 0.74 NPC1 (0.43) AKT1AKT2NPC1RAB9AMAPK10
SCHEMBL31190884 0.74 MAPK10 (0.56) AKT1AKT2NPC1RAB9AMAPK10
SCHEMBL31190927 0.73 CGAS (0.40) AKT1AKT2NPC1RAB9ASMN1; SMN2
SCHEMBL31190886 0.73 AKT1 (0.42) AKT1AKT2NPC1RAB9ASMN1; SMN2
SCHEMBL31091889 0.72 AKT1 (0.41) AKT1AKT2NPC1RAB9ASMN1; SMN2
SCHEMBL31091944 0.72 AKT1 (0.43) AKT1AKT2NPC1RAB9ASMN1; SMN2
SCHEMBL31190889 0.71 GRM2 (0.42) AKT1AKT2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024220543-A1 NK3 MODULATORS AND USES THEREOF KALLYOPE, INC. (US) 2024-10-24 WO disclosed