SCHEMBL3126629

SCHEMBL3126629

NC(=O)CCCc1cncc(S(N)(=O)=O)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.49
CA2 P00918 15/20 0.39
CA1 P00915 8/20 0.38
CA12 O43570 5/20 0.36
CA9 Q16790 4/20 0.36
CA6 P23280 3/20 0.36
CA7 P43166 3/20 0.36
CA4 P22748 2/20 0.36
CA5A P35218 2/20 0.36
CA14 Q9ULX7 2/20 0.36
CA5B Q9Y2D0 2/20 0.36
CA13 Q8N1Q1 2/20 0.36
CA3 P07451 1/20 0.36
TLR8 Q9NR97 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FAAH O00519 1/20 0.35
CES1 P23141 1/20 0.35
TBXAS1 P24557 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313325 0.86 CYP11B2 (0.37) APLNRTBXAS1
SCHEMBL4304457 0.82 CA2 (0.42) CA2TBXAS1
SCHEMBL3132047 0.82 ALDH1A1 (0.39) SMN1; SMN2TBXAS1
SCHEMBL24883427 0.76 APLNR (0.58) APLNRCA2CA1CA12CA9
SCHEMBL4306556 0.76 KDM4E (0.45) SMN1; SMN2
SCHEMBL2433226 0.76 HCAR2 (0.42) SMN1; SMN2TBXAS1
SCHEMBL9978250 0.74 APLNR (0.55) APLNRCA2CA1CA12CA9
SCHEMBL4316426 0.74 PIK3CB (0.46) SMN1; SMN2
SCHEMBL27940556 0.73 APLNR (0.46) APLNRCA2CA1CA12CA9
SCHEMBL24883515 0.73 APLNR (0.53) APLNRCA2CA1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036632-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed