SCHEMBL31293675

SCHEMBL31293675

CN(C)Cc1ccc(NC(=O)NC2CC3(C2)CN(C(=O)c2cnn4ccsc24)C3)cc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 7/20 0.43
CCNC P24863 6/20 0.43
EPHX2 P34913 11/20 0.38
RET P07949 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31293664 0.89 CDK8 (0.47) CDK8CCNCRET
SCHEMBL31293875 0.83 EPHX2 (0.46) CDK8EPHX2
SCHEMBL31293436 0.81 UBE2M (0.35) EPHX2
SCHEMBL31293851 0.80 SCN10A (0.35) EPHX2KDR
SCHEMBL31293858 0.80 KMT2A (0.43) EPHX2
SCHEMBL31293631 0.79 EPHX2 (0.43) EPHX2KDR
SCHEMBL31293410 0.79 ENPP2 (0.35) EPHX2
SCHEMBL31293883 0.78 CDK8 (0.45) CDK8CCNCEPHX2RETKDR
SCHEMBL31293519 0.78 RAB9A (0.46) CDK8CCNCEPHX2
SCHEMBL31293478 0.77 SYK (0.39) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724439-A1 HETEROARYL DERIVATIVES AS DDRS INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2026-04-15 EP claimed
WO-2024251855-A1 HETEROARYL DERIVATIVES AS DDRS INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2024-12-12 WO claimed