SCHEMBL3129552

SCHEMBL3129552

COc1ccc(NCc2cncs2)cc1OC(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPX4 P36969 12/20 0.43
MAPT P10636 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 2/20 0.40
GLA P06280 1/20 0.40
CASP1 P29466 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRM4 Q14833 1/20 0.40
PDE4B Q07343 1/20 0.39
LMNA P02545 2/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AAK1 Q2M2I8 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3118114 0.92 CYP3A4 (0.39) GPX4PDE4BLMNASMN1; SMN2AAK1
SCHEMBL3207727 0.89 CYP2C19 (0.39) GPX4MAPTMEN1KMT2APDE4B
SCHEMBL3121001 0.89 GPX4 (0.44) GPX4MAPTMEN1KMT2AKDM4E
SCHEMBL3128380 0.82 KDM4E (0.50) GPX4MAPTMEN1KMT2AKDM4E
SCHEMBL3126018 0.80 DHFR (0.48) GPX4MAPTMEN1KMT2AKDM4E
SCHEMBL3120371 0.80 AAK1 (0.41) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL3118081 0.78 PDE4B (0.41) GPX4MAPTMEN1KMT2AKDM4E
SCHEMBL3129215 0.77 L3MBTL1 (0.56) MAPTMEN1KMT2AALDH1A1GAA
SCHEMBL3131820 0.77 GRM4 (0.44) GPX4MAPTMEN1KMT2AKDM4E
SCHEMBL2908810 0.76 EGFR (0.45) GPX4MAPTKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010003084-A2 PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2010-01-07 WO disclosed