SCHEMBL31320118

SCHEMBL31320118

CCNC(=O)Nc1ncnc(Cl)c1F

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.41
KDR P35968 2/20 0.41
EGFR P00533 4/20 0.41
ERBB2 P04626 3/20 0.41
SIGMAR1 Q99720 2/20 0.40
FGFR1 P11362 2/20 0.37
SRC P12931 2/20 0.37
FGFR2 P21802 1/20 0.37
FGFR4 P22455 1/20 0.37
FGFR3 P22607 1/20 0.37
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31032943 0.82 SIGMAR1 (0.41) ABL1KDREGFRERBB2SIGMAR1
SCHEMBL31032965 0.81 KDR (0.41) ABL1KDREGFRERBB2SIGMAR1
SCHEMBL1439729 0.79 KDM4E (0.40) EGFR
SCHEMBL31032954 0.78 GAA (0.43) ABL1KDREGFRERBB2SIGMAR1
SCHEMBL31320113 0.76 KDR (0.36) ABL1KDREGFRERBB2SIGMAR1
SCHEMBL23396651 0.73 MAPT (0.31)
SCHEMBL31320125 0.71 ABL1 (0.44) ABL1FGFR1SRCJAK2JAK1
SCHEMBL31320131 0.70 ABL1 (0.44) ABL1FGFR1SRCJAK2JAK1
SCHEMBL1440229 0.69 PDPK1 (0.37) TYK2
SCHEMBL31320136 0.69 GAA (0.51) ABL1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024240108-A1 ARYL UREA PARP1 INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF 上海海和药物研究开发股份有限公司 2024-11-28 WO disclosed