SCHEMBL31320113

SCHEMBL31320113

CCNC(=O)Nc1ncnc(COS(C)(=O)=O)c1F

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.36
ABL1 P00519 3/20 0.36
SIGMAR1 Q99720 2/20 0.35
EGFR P00533 3/20 0.34
ERBB2 P04626 3/20 0.34
GAA P10253 1/20 0.33
MKNK2 Q9HBH9 2/20 0.32
BRAF P15056 2/20 0.32
MKNK1 Q9BUB5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31032965 0.80 KDR (0.41) KDRABL1SIGMAR1EGFRERBB2
SCHEMBL31032943 0.79 SIGMAR1 (0.41) KDRABL1SIGMAR1EGFRERBB2
SCHEMBL31320118 0.76 ABL1 (0.41) KDRABL1SIGMAR1EGFRERBB2
SCHEMBL31032954 0.73 GAA (0.43) KDRABL1SIGMAR1EGFRERBB2
SCHEMBL31320136 0.67 GAA (0.51) KDRABL1GAA
SCHEMBL31320125 0.63 ABL1 (0.44) ABL1MKNK2
SCHEMBL28821088 0.63 TGFBR1 (0.36) GAA
SCHEMBL15164126 0.63 CYP1A2 (0.31)
SCHEMBL31320131 0.62 ABL1 (0.44) ABL1MKNK2
SCHEMBL13632472 0.62 ABL1 (0.40) KDRABL1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024240108-A1 ARYL UREA PARP1 INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF 上海海和药物研究开发股份有限公司 2024-11-28 WO disclosed