SCHEMBL3133

SCHEMBL3133

CC(C)[C@H](NCc1ccc(-c2ccccc2C#N)cc1Br)C(=O)OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 12/20 0.43
CD274 Q9NZQ7 12/20 0.43
FFAR1 O14842 2/20 0.39
AKR1B1 P15121 1/20 0.39
CTSL P07711 2/20 0.39
CTSB P07858 2/20 0.39
CTSK P43235 2/20 0.39
CTSS P25774 1/20 0.39
ADAMTS4 O75173 1/20 0.38
MMP13 P45452 1/20 0.38
PTPN1 P18031 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2317 0.85 FFAR1 (0.48) FFAR1AKR1B1CTSLCTSBCTSK
SCHEMBL14004740 0.85 FFAR1 (0.48) FFAR1AKR1B1CTSLCTSBCTSK
Hydrochloric Acid SCHEMBL2728 0.84 FFAR1 (0.47) FFAR1AKR1B1CTSLCTSBCTSK
Hydrochloric Acid SCHEMBL3473569 0.84 FFAR1 (0.47) FFAR1AKR1B1CTSLCTSBCTSK
SCHEMBL8813467 0.84 FFAR1 (0.44) PDCD1CD274FFAR1AKR1B1CTSL
SCHEMBL2437416 0.79 CTSS (0.42) CD274CTSLCTSBCTSKCTSS
SCHEMBL14032424 0.78 FFAR1 (0.47) FFAR1AKR1B1CTSLCTSBCTSK
SCHEMBL2780 0.78 FFAR1 (0.35) FFAR1AKR1B1CTSLCTSBCTSK
Hydrochloric Acid SCHEMBL3412065 0.78 CTSB (0.41) CD274CTSLCTSBCTSKCTSS
SCHEMBL2779 0.77 AGTR1 (0.42) FFAR1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed