SCHEMBL3133401

SCHEMBL3133401

N#Cc1ccc2[nH]c(OC(=O)O)cc2n1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.37
PIN1 Q13526 1/20 0.37
MAPK10 P53779 4/20 0.35
ENPP1 P22413 2/20 0.33
MET P08581 2/20 0.33
CAMKK2 Q96RR4 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
CHEK2 O96017 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
AHR P35869 1/20 0.30
SRC P12931 1/20 0.30
CTSB P07858 1/20 0.30
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3141851 0.78 CAMKK2 (0.35) NQO1PIN1CAMKK2SRCCTSB
SCHEMBL3128146 0.78 GRIN2D (0.35) RAB9AMAPT
SCHEMBL3140892 0.78 HDAC6 (0.33) HDAC6MAPT
SCHEMBL2107950 0.78 SMAD3 (0.45) PIN1MAPTKMT2AAHR
SCHEMBL3412763 0.77 CYP19A1 (0.50) PIN1CYP19A1
SCHEMBL3145657 0.75 CHEK1 (0.38) PIN1ENPP1
SCHEMBL3136953 0.75 POLB (0.40) ENPP1HDAC6MAPTKMT2A
SCHEMBL3127269 0.74 CHEK1 (0.37) PIN1ENPP1
SCHEMBL15567755 0.73 GABRP (0.39) NPC1RAB9AMAPT
SCHEMBL22533604 0.70 NQO1 (0.44) NQO1METMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636224-B1 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDE INHIBITORS OF GLYCOGEN PHOSHORYLASE PROSIDION LTD (GB) 2010-07-14 EP claimed