SCHEMBL3145657

SCHEMBL3145657

N#Cc1cc2cc(OC(=O)O)[nH]c2cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 13/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRB2 P47870 1/20 0.37
GABRA4 P48169 1/20 0.37
GABRE P78334 1/20 0.37
GABRA6 Q16445 1/20 0.37
GABRG1 Q8N1C3 1/20 0.37
GABRG3 Q99928 1/20 0.37
GABRQ Q9UN88 1/20 0.37
ENPP1 P22413 3/20 0.33
PIN1 Q13526 1/20 0.32
PDPK1 O15530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3127269 0.90 CHEK1 (0.37) CHEK1GABRPGABRDGABRA1GABRB1
SCHEMBL3141184 0.87 GABRA1 (0.30) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL3138608 0.79 CHEK1 (0.41) CHEK1GABRPGABRDGABRA1GABRB1
SCHEMBL3137099 0.79 NR3C1 (0.34) PIN1
SCHEMBL3136216 0.79
SCHEMBL2107455 0.77 GPR35 (0.49) CHEK1GABRPGABRDGABRA1GABRB1
SCHEMBL3133401 0.75 NQO1 (0.37) ENPP1PIN1
SCHEMBL3412763 0.75 CYP19A1 (0.50) PIN1
SCHEMBL3141851 0.73 CAMKK2 (0.35) CHEK1PIN1PDPK1DYRK3MAP4K4
SCHEMBL4038601 0.71 DAO (0.51) CSNK2A1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636224-B1 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDE INHIBITORS OF GLYCOGEN PHOSHORYLASE PROSIDION LTD (GB) 2010-07-14 EP claimed