SCHEMBL3136953

SCHEMBL3136953

COc1ccc2[nH]c(OC(=O)O)cc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
MTNR1A P48039 3/20 0.36
MTNR1B P49286 3/20 0.36
ENPP3 O14638 1/20 0.36
ENPP1 P22413 1/20 0.36
ENPP2 Q13822 1/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
NNMT P40261 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12614229 0.82 SIRT2 (0.46) SIRT2SIRT1MTNR1AMTNR1BENPP3
SCHEMBL3140892 0.82 HDAC6 (0.33) KDM4EL3MBTL1ADORA2AADORA1MAPT
SCHEMBL15567755 0.80 GABRP (0.39) ALDH1A1KDM4EL3MBTL1CYP1A2CYP2C19
SCHEMBL3128146 0.79 GRIN2D (0.35) POLBSIRT2ALDH1A1KDM4EMAPT
SCHEMBL2107849 0.79 PIN1 (0.47) POLBTDP1SIRT2SIRT1MTNR1A
SCHEMBL30310720 0.79 PIN1 (0.47) POLBTDP1SIRT2SIRT1MTNR1A
SCHEMBL3133401 0.75 NQO1 (0.37) ENPP1MAPTKMT2AHDAC6
SCHEMBL30310722 0.75 NNMT (0.46) POLBTDP1SIRT2SIRT1MTNR1A
SCHEMBL3754482 0.75 XDH (0.47) SIRT2SIRT1MTNR1AMTNR1BALDH1A1
SCHEMBL4034495 0.75 NNMT (0.46) POLBTDP1SIRT2SIRT1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636224-B1 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDE INHIBITORS OF GLYCOGEN PHOSHORYLASE PROSIDION LTD (GB) 2010-07-14 EP claimed