SCHEMBL3133992

SCHEMBL3133992

O=[N+]([O-])C(CO)c1ccnc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.36
IDO1 P14902 2/20 0.33
MAPT P10636 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
THRB P10828 1/20 0.33
PKM P14618 1/20 0.33
RECQL P46063 1/20 0.33
TDO2 P48775 1/20 0.33
BLM P54132 1/20 0.33
CASP6 P55212 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GSR P00390 1/20 0.32
CTSA P10619 1/20 0.32
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1028353 0.76 ALDH1A1 (0.49) LOXL2IDO1MAPTTDP1KDM4E
SCHEMBL4298042 0.74 CES2 (0.36) GSR
SCHEMBL3336779 0.70 GSR (0.55) MAPTTDP1KDM4EMEN1ALDH1A1
SCHEMBL6511267 0.69 PTGDR2 (0.41) LOXL2KDM4EMEN1ALDH1A1PKM
SCHEMBL16463407 0.69 TRPV4 (0.40)
Fluoride SCHEMBL28046654 0.68 GSR (0.53) MAPTTDP1KDM4EMEN1ALDH1A1
SCHEMBL4851936 0.68 ALDH1A1 (0.47) MAPTTDP1MEN1ALDH1A1LMNA
SCHEMBL25356422 0.67 LOXL2 (0.50) LOXL2MAPTTDP1KDM4EMEN1
SCHEMBL6258107 0.67 ALDH1A1 (0.53) LOXL2IDO1MAPTTDP1KDM4E
SCHEMBL2461283 0.67 IGF1R (0.37) MAPTKDM4EMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150546-A2 PYRIMIDINE DERIVATIVES AS INHIBITORS OF PHOSPHATIDYLINOSITOL-3-KINASE F. Hoffmann-Roche AG (CH) 2010-02-10 EP disclosed
WO-2008125839-A2 PYRIMIDINE DERIVATIVES AS INHIBITORS OF PHOSPHATIDYLINOSITOL-3-KINASE PIRAMED LIMITED (GB) 2008-10-23 WO disclosed