SCHEMBL3137034

SCHEMBL3137034

CNC1(COc2cncc(-c3cc(Cl)cc(Cl)c3)c2)CC1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
INPPL1 O15357 2/20 0.41
CHRNB2 P17787 4/20 0.37
CHRNB1 P11230 2/20 0.37
CHRNB4 P30926 2/20 0.37
CHRNA3 P32297 2/20 0.37
CHRNB3 Q05901 2/20 0.37
CHRNA4 P43681 2/20 0.35
AKT1 P31749 1/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3145280 0.88 CHRNB1 (0.49) INPPL1CHRNB2CHRNB1CHRNB4CHRNA3
SCHEMBL3147306 0.88 INPPL1 (0.43) INPPL1CHRNB2CHRNB1CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL3151937 0.87 CHRNB1 (0.48) INPPL1CHRNB2CHRNB1CHRNB4CHRNA3
SCHEMBL3143138 0.84 INPPL1 (0.39) INPPL1
SCHEMBL3147229 0.83 CHRNB2 (0.49) INPPL1CHRNB2CHRNB1CHRNB4CHRNA3
SCHEMBL3150890 0.83 INPPL1 (0.46) INPPL1CHRNB2CHRNB1CHRNB4CHRNA3
SCHEMBL3141790 0.82 CHRNB2 (0.48) INPPL1CHRNB2CHRNB1CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL3765553 0.82 CHRNB2 (0.48) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3
SCHEMBL3150832 0.81 ACVR1B (0.40) CYP1A1CYP1B1
SCHEMBL3150922 0.81 CHRNB1 (0.49) INPPL1CHRNB2CHRNB1CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed