Carbimazole

Carbimazole

SCHEMBL3137059

CCOC(=O)n1ccn(C)c1=S.[NaH].[NaH]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TPO

The experimentally established mechanism targets of Carbimazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LPO P22079 9/20 0.96
LMNA P02545 1/20 0.96
CYP1A2 P05177 1/20 0.96
BCHE P06276 1/20 0.36
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
BAZ2B Q9UIF8 1/20 0.33
BAZ2A Q9UIF9 1/20 0.33
TSHR P16473 2/20 0.33
GSK3B P49841 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
GSK3A P49840 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbimazole SCHEMBL44211 0.98 LPO (1.00) LPOLMNACYP1A2BCHEALDH1A1
Carbimazole SCHEMBL28078672 0.96 LPO (0.96) LPOLMNACYP1A2BCHEALDH1A1
Carbimazole SCHEMBL28086764 0.85 LPO (0.75) LPOLMNACYP1A2BCHEALDH1A1
Carbimazole SCHEMBL20771744 0.80 LPO (0.66) LPOLMNACYP1A2ALDH1A1TSHR
SCHEMBL26295022 0.71 LPO (0.57) LPOLMNACYP1A2BCHEALDH1A1
SCHEMBL7548705 0.66 LPO (0.50) LPOLMNACYP1A2BCHEALDH1A1
SCHEMBL15284133 0.66 LPO (0.50) LPOLMNACYP1A2BCHEALDH1A1
SCHEMBL29117082 0.64 LPO (0.49) LPOLMNACYP1A2BCHEALDH1A1
SCHEMBL13278237 0.64 LPO (0.49) LPOLMNACYP1A2BCHEALDH1A1
SCHEMBL163149 0.63 LPO (0.47) LPOLMNACYP1A2BCHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2203192-A1 WOUND CARE FORMULATION Northern Health And Social Care Trust (GB) 2010-07-07 EP disclosed
WO-2009037500-A1 WOUND CARE FORMULATION NORTHERN HEALTH AND SOCIAL CARE TRUST (GB) 2009-03-26 WO disclosed