SCHEMBL31385169

SCHEMBL31385169

Cc1nc(C(=O)NC(C)c2ccccn2)c2ccccc2n1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 11/20 0.53
ADORA2B P29275 4/20 0.53
ADORA3 P0DMS8 2/20 0.53
PARP1 P09874 2/20 0.52
PARP3 Q9Y6F1 1/20 0.52
PPARG P37231 1/20 0.46
TACR3 P29371 2/20 0.45
CHRM4 P08173 1/20 0.44
SSTR4 P31391 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31385143 0.83 TACR3 (0.57) ADORA2AADORA2BTACR3
SCHEMBL31385144 0.81 ROCK2 (0.55) ADORA2AADORA2BPPARGTACR3
SCHEMBL31385239 0.80 TACR3 (0.51) ADORA3TACR3
SCHEMBL31385233 0.78 ADORA2B (0.53) ADORA2AADORA2BADORA3TACR3CHRM4
SCHEMBL14094521 0.78 TACR3 (0.60) ADORA2ATACR3
SCHEMBL6392481 0.78 PARP1 (0.49) ADORA2AADORA2BADORA3PARP1PARP3
SCHEMBL31385183 0.78 ADORA2A (0.48) ADORA2APPARGTACR3SSTR4
SCHEMBL31385131 0.78 MAOA (0.61) TACR3
SCHEMBL14094516 0.76 TACR3 (0.75) TACR3
SCHEMBL31385130 0.76 PTGER4 (0.56) ADORA3TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119119035-A RIPK1 kinase target inhibitor and preparation method and application thereof 中山大学 2024-12-13 CN disclosed