SCHEMBL31385183

SCHEMBL31385183

Cc1nc(C(=O)NC(C)c2ccccc2F)c2ccccc2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
PPARG P37231 1/20 0.44
TACR3 P29371 3/20 0.43
KMT2A Q03164 2/20 0.43
CYP2C9 P11712 2/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ROCK2 O75116 6/20 0.43
ROCK1 Q13464 6/20 0.43
SSTR4 P31391 1/20 0.42
HSD17B13 Q7Z5P4 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31385143 0.83 TACR3 (0.57) ADORA2ATACR3CYP2C9CYP1A2CYP3A4
SCHEMBL31385131 0.82 MAOA (0.61) TACR3KMT2ACYP2C9MEN1CYP1A2
SCHEMBL31385140 0.80 GAA (0.55) PPARGTACR3CYP2C9CYP1A2CYP3A4
SCHEMBL31385239 0.80 TACR3 (0.51) TACR3KMT2ACYP2C9MEN1CYP1A2
SCHEMBL31385144 0.79 ROCK2 (0.55) ADORA2APPARGTACR3KMT2ACYP2C9
SCHEMBL28049266 0.78 NPC1 (0.58) PPARGKMT2ACYP2C9MEN1CYP1A2
SCHEMBL31385169 0.78 ADORA2A (0.53) ADORA2APPARGTACR3SSTR4
SCHEMBL25375819 0.76 GAA (0.50) PPARGKMT2AMEN1ROCK2ROCK1
SCHEMBL31385130 0.76 PTGER4 (0.56) TACR3KMT2AMEN1MAPT
SCHEMBL31385233 0.76 ADORA2B (0.53) ADORA2AADORA1TACR3CYP2C9ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119119035-A RIPK1 kinase target inhibitor and preparation method and application thereof 中山大学 2024-12-13 CN disclosed