SCHEMBL31405

SCHEMBL31405

COc1cc(C(=O)c2nc3ccccc3s2)ccc1F

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 3/20 0.70
HSD17B2 P37059 3/20 0.70
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 3/20 0.52
HTT P42858 3/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2B6 P20813 1/20 0.52
CYP2C19 P33261 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52
TUBB3 Q13509 1/20 0.52
TUBB2A Q13885 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30222 0.86 HSD17B1 (0.79) HSD17B1HSD17B2HTTCYP1A2CYP3A4
SCHEMBL427929 0.84 TUBB4A (0.72) HSD17B1HSD17B2ALDH1A1KDM4EHTT
SCHEMBL22526 0.82 HSD17B1 (1.00) HSD17B1HSD17B2ALDH1A1CYP1A2CYP3A4
SCHEMBL11007700 0.79 KMT2A (0.66) HSD17B1HSD17B2ALDH1A1KDM4EHTT
SCHEMBL31078 0.79 RAB9A (0.65) HSD17B1HSD17B2ALDH1A1KDM4EMEN1
SCHEMBL4088536 0.77 HSD17B1 (0.68) HSD17B1HSD17B2ALDH1A1KDM4EHTT
SCHEMBL14021104 0.77 RAB9A (0.62) ALDH1A1KDM4EHTTL3MBTL1MEN1
SCHEMBL27623260 0.76 HSD17B1 (0.67) HSD17B1HSD17B2ALDH1A1CYP1A2CYP3A4
SCHEMBL28094523 0.75 CYP1A2 (0.68) ALDH1A1HTTCYP1A2CYP3A4CYP2D6
SCHEMBL27246607 0.75 HSD17B1 (0.60) HSD17B1HSD17B2HTTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed