SCHEMBL22526

SCHEMBL22526

O=C(c1ccc(F)c(O)c1)c1nc2ccccc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 9/20 1.00
HSD17B2 P37059 8/20 1.00
CYP1A2 P05177 2/20 0.74
CYP3A4 P08684 2/20 0.74
CYP2D6 P10635 2/20 0.74
CYP2C9 P11712 2/20 0.74
CYP2B6 P20813 2/20 0.74
CYP2C19 P33261 2/20 0.74
HSD17B14 Q9BPX1 5/20 0.56
BCL2 P10415 1/20 0.50
MCL1 Q07820 1/20 0.50
BAD Q92934 1/20 0.50
TOP1 P11387 2/20 0.49
CLK1 P49759 1/20 0.49
DYRK1A Q13627 1/20 0.49
DYRK1B Q9Y463 1/20 0.49
ALPL P05186 1/20 0.48
ALPG P10696 1/20 0.48
GCGR P47871 1/20 0.48
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29673 0.85 HSD17B1 (1.00) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL31405 0.82 HSD17B1 (0.70) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL4088536 0.81 HSD17B1 (0.68) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL30687 0.80 HSD17B1 (1.00) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL27623260 0.80 HSD17B1 (0.67) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL1304947 0.80 HSD17B1 (0.66) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL31407 0.79 HSD17B1 (0.79) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL14020417 0.79 HSD17B1 (0.64) HSD17B1HSD17B2BCL2MCL1BAD
SCHEMBL24751 0.78 HSD17B1 (0.62) HSD17B1HSD17B2BCL2MCL1BAD
SCHEMBL6319718 0.77 ALDH1A1 (0.66) HSD17B1HSD17B2MCL1DYRK1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP claimed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO claimed
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed