SCHEMBL315779

SCHEMBL315779

CN(C)C1(Cc2ccc(Cl)cc2)CCC(NC(=O)c2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.44
TRPC3 Q13507 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 3/20 0.42
SPR P35270 1/20 0.42
DDR1 Q08345 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
DDR2 Q16832 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
MAP3K20 Q9NYL2 1/20 0.41
MAP3K2 Q9Y2U5 1/20 0.41
GPR6 P46095 1/20 0.41
CRHR1 P34998 1/20 0.41
CCR1 P32246 3/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315130 0.97 NPC1 (0.45) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL316498 0.97 NPSR1 (0.44) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL315976 0.96 KDM4E (0.48) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL315879 0.92 CCR1 (0.44) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL316470 0.88 KDM4E (0.43) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL315268 0.88 ALDH1A1 (0.43) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL315441 0.88 KDM4E (0.46) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL10366974 0.84 HSD11B1 (0.56) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL2851938 0.82 SPR (0.56) HSD11B1TRPC3KDM4EALDH1A1MAPT
SCHEMBL2854286 0.79 HSD11B1 (0.52) HSD11B1TRPC3KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed