SCHEMBL3157490

SCHEMBL3157490

CC(=O)NC(N)CCCBr

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.34
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM1 P11229 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
THRB P10828 1/20 0.32
ALOX15 P16050 1/20 0.32
NFKB1 P19838 1/20 0.32
PTGS2 P35354 1/20 0.32
THPO P40225 1/20 0.32
RECQL P46063 1/20 0.32
BLM P54132 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GNPAT O15228 1/20 0.32
ALDH1A1 P00352 1/20 0.31
SIRT6 Q8N6T7 1/20 0.31
SIRT1 Q96EB6 1/20 0.31
PLA2G2C Q5R387 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7520216 0.92 TRPV1 (0.40) TRPV1CHRM2CHRM4CHRM1KDM4E
SCHEMBL12478006 0.81 PLA2G2C (0.46) SIRT6SIRT1PLA2G2C
SCHEMBL17213387 0.79 SIRT6 (0.47) SIRT6SIRT1PLA2G2C
SCHEMBL7801151 0.78 SIRT6 (0.50) TRPV1SIRT6SIRT1
SCHEMBL7085362 0.76
Benzene SCHEMBL9177693 0.73 SIRT6 (0.43) MAPTALDH1A1SIRT6SIRT1PLA2G2C
SCHEMBL5596648 0.72 GABRP (0.52) MAPTNFKB1BLMGNPATPLA2G2C
SCHEMBL28663197 0.72 MTNR1A (0.41) ALDH1A1
SCHEMBL24158519 0.72 ALOX15 (0.37) KDM4EALOX15SMN1; SMN2SIRT6SIRT1
SCHEMBL20892574 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497525-B2 Pneumococcal polysaccharide conjugate vaccine MERCK & CO INC (US) 2010-03-03 EP disclosed
EP-0497525-B1 Pneumococcal polysaccharide conjugate vaccine MERCK & CO INC (US) 1998-08-19 EP disclosed
US-5623057-A IMMUNOGENIC PROTEIN COVALENTLY LINKED TO POLYSACCHARIDE DERIVED FROM STREPTOCOCCUS PNEUMONIAE MERCK & CO., INC. (US) 1997-04-22 US disclosed
US-5371197-A Protein-dimeric polysaccharide conjugate vaccine MERCK & CO., INC. (US) 1994-12-06 US disclosed
EP-0534764-A1 Protein-dimeric polysaccharide conjugate vaccine MERCK & CO. INC. (US) 1993-03-31 EP disclosed
EP-0497525-A2 Pneumococcal polysaccharide conjugate vaccine MERCK & CO. INC. (US) 1992-08-05 EP disclosed
EP-0186576-B1 COVALENTLY-MODIFIED NEUTRAL BACTERIAL POLYSACCHARIDES, STABLE COVALENT CONJUGATES OF SUCH POLYSACCHARIDES AND IMMUNOGENIC PROTEINS, AND METHODS OF PREPARING SUCH POLYSACCHARIDES AND CONJUGATES MERCK & CO. INC. (US) 1992-07-22 EP disclosed
EP-0467714-A1 The class II protein of the outer membrane of neisseria meningitidis MERCK & CO. INC. (US) 1992-01-22 EP disclosed
EP-0161188-B1 COVALENTLY-MODIFIED BACTERIAL POLYSACCHARIDES, STABLE COVALENT CONJUGATES OF SUCH POLYSACCHARIDES AND IMMUNOGENIC PROTEINS WITH BIGENERIC SPACERS, AND METHODS OF PREPARING SUCH POLYSACCHARIDES AND CONJUGATES AND OF CONFIRMING COVALENCY MERCK & CO. INC. (US) 1991-04-03 EP disclosed
US-4882317-A SOLUBILIZATION MERCK & CO., INC. (US) 1989-11-21 US disclosed
US-4830852-A COVALENT-MODIFICATION AND HAVING A COUPLING SPACER CONTAINING A THIOETHER; VACCINES; CHEMICAL STABILITY; INFANT PROTECTION MERCK & CO INC. (US) 1989-05-16 US disclosed
US-4695624-A Covalently-modified polyanionic bacterial polysaccharides, stable covalent conjugates of such polysaccharides and immunogenic proteins with bigeneric spacers, and methods of preparing such polysaccharides and conjugates and of confirming covalency MERCK & CO., INC. (US) 1987-09-22 US disclosed
EP-0186576-A2 Covalently-modified neutral bacterial polysaccharides, stable covalent conjugates of such polysaccharides and immunogenic proteins, and methods of preparing such polysaccharides and conjugates MERCK & CO. INC. (US) 1986-07-02 EP disclosed
EP-0161188-A2 Covalently-modified bacterial polysaccharides, stable covalent conjugates of such polysaccharides and immunogenic proteins with bigeneric spacers, and methods of preparing such polysaccharides and conjugates and of confirming covalency MERCK & CO. INC. (US) 1985-11-13 EP disclosed