SCHEMBL3170868

SCHEMBL3170868

COc1ccc(CC(=O)NCCNc2cc(NCCNC(C)=O)nc(-c3ccc(Cl)cc3)n2)cc1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.49
CA2 P00918 2/20 0.45
CA1 P00915 1/20 0.45
TP53 P04637 2/20 0.43
IARS1 P41252 1/20 0.43
GAA P10253 2/20 0.41
KDR P35968 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.39
CETP P11597 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3177128 0.93 LMNA (0.49) LMNACA2CA1TP53IARS1
SCHEMBL3163050 0.91 BCHE (0.45) CA2CA1TP53IARS1GAA
SCHEMBL3162053 0.89 LMNA (0.49) LMNACA2CA1TP53IARS1
SCHEMBL3176265 0.87 MEN1 (0.50) TP53KDRADORA3
SCHEMBL3171330 0.84 CA1 (0.48) LMNACA2CA1TP53
SCHEMBL3164379 0.84 TP53 (0.52) LMNATP53GAAKDRADORA3
SCHEMBL3172113 0.83 CSNK1D (0.47) LMNATP53GAA
SCHEMBL3171164 0.83 MTNR1A (0.49) CA2CA1IARS1GAA
SCHEMBL3162657 0.83 CETP (0.43) LMNATP53GAACETP
SCHEMBL3169166 0.83 ALDH1A1 (0.49) LMNATP53ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465631-B1 PYRIMIDINE A2B SELECTIVE ANTAGONIST COMPOUNDS, THEIR SYNTHESIS AND USE OSI PHARM INC (US) 2010-02-24 EP disclosed