SCHEMBL3174797

SCHEMBL3174797

O=C(O)CCCC(Cc1ccccc1)C(=O)O

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPA3 P15088 3/20 0.80
FOLH1 Q04609 2/20 0.70
CYP1A2 P05177 1/20 0.66
CPA1 P15085 2/20 0.62
CPB1 P15086 1/20 0.62
CPB2 Q96IY4 1/20 0.62
NAALAD2 Q9Y3Q0 1/20 0.55
LTA4H P09960 1/20 0.54
HDAC3 O15379 1/20 0.53
MAPK1 P28482 1/20 0.53
ADRA1A P35348 1/20 0.53
HDAC4 P56524 1/20 0.53
SLC6A3 Q01959 1/20 0.53
HDAC1 Q13547 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC2 Q92769 1/20 0.53
HDAC10 Q969S8 1/20 0.53
HDAC11 Q96DB2 1/20 0.53
HDAC8 Q9BY41 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12494537 1.00 CPA3 (0.80) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL26679347 0.95 CPA3 (0.77) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL28430963 0.93 CPA3 (0.75) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL31303730 0.93 CPA3 (0.75) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL11143841 0.93 CPA3 (0.75) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL28600681 0.93 CPA3 (0.75) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL29088272 0.89 CPA3 (1.00) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL3963424 0.89 CPA3 (1.00) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL11664393 0.89 FOLH1 (0.79) CPA3FOLH1CYP1A2CPA1CPB1
SCHEMBL22612309 0.86 FOLH1 (0.71) CPA3FOLH1CYP1A2CPA1CPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4700124-A2 OLIGONUCLEOTIDE-LIGAND CONJUGATES AND PROCESS FOR THEIR PREPARATION Alnylam Pharmaceuticals, Inc. (US) 2026-02-25 EP disclosed
US-20250326731-A1 CATALYST-CONTROLLED SITE-SELECTIVE METHYLENE C-H LACTONIZATION OF DICARBOXYLIC ACIDS SCRIPPS RESEARCH INST (US) 2025-10-23 US disclosed
EP-4522595-A2 CATALYST-CONTROLLED SITE-SELECTIVE METHYLENE C-H LACTONIZATION OF DICARBOXYLIC ACIDS The Scripps Research Institute (US) 2025-03-19 EP disclosed
US-20250075208-A1 OLIGONUCLEOTIDE-LIGAND CONJUGATES AND PROCESS FOR THEIR PREPARATION BANK OF AMERICA, N.A. 2025-03-06 US disclosed
US-12173288-B2 Oligonucleotide-ligand conjugates and process for their preparation ALNYLAM PHARMACEUTICALS, INC. (US) 2024-12-24 US disclosed
WO-2023220559-A2 CATALYST-CONTROLLED SITE-SELECTIVE METHYLENE C-H LACTONIZATION OF DICARBOXYLIC ACIDS THE SCRIPPS RESEARCH INSTITUTE (US) 2023-11-16 WO disclosed
WO-2023220559-A2 CATALYST-CONTROLLED SITE-SELECTIVE METHYLENE C-H LACTONIZATION OF DICARBOXYLIC ACIDS THE SCRIPPS RESEARCH INSTITUTE (US) 2023-11-16 WO disclosed
US-20220348914-A1 OLIGONUCLEOTIDE-LIGAND CONJUGATES AND PROCESS FOR THEIR PREPARATION BANK OF AMERICA, N.A. 2022-11-03 US disclosed
EP-4039278-A1 OLIGONUCLEOTIDE-LIGAND CONJUGATES AND PROCESS FOR THEIR PREPARATION Alnylam Pharmaceuticals, Inc. (US) 2022-08-10 EP disclosed
EP-3019200-B1 OLIGONUCLEOTIDE-LIGAND CONJUGATES AND PROCESS FOR THEIR PREPARATION ALNYLAM PHARMACEUTICALS INC (US) 2022-03-23 EP disclosed
US-6262195-B1 POLYMERIZING ETHYLENE OPTIONALLY WITH ALPHA-OLEFIN IN PRESENCE OF TITANIUM OR VANADIUM COMPOUND CATALYST; CONTACTING PRODUCT WITH COMPOUND TO DEACTIVATE CATALYST, ZIRCOCENE CATALYST AND COCATALYST TO FURTHER POLYMERIZE MONTELL TECHNOLOGY COMPANY BV (NL) 2001-07-17 US disclosed
US-6232484-B1 Bridged zirconocene compounds, process for their preparation and their use as catalyst components in the polymerization of olefins MONTELL TECHNOLOGY B.V. (NL) 2001-05-15 US disclosed
EP-0941997-A2 Bridged zirconocene compounds, process for their preparation, and their use as catalyst components in the polymerization of olefins Montell Technology Company bv (NL) 1999-09-15 EP disclosed
EP-0942011-A1 Multi-stage process for the polymerization of olefins Montell Technology Company bv (NL) 1999-09-15 EP disclosed
US-5911995-A ENZYME INHIBITORS FOR TYROSINE KINASE AND CYTOTOXIC DOSAGE OF EPIDERMAL GROWTH FACTOR REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1999-06-15 US disclosed
WO-1997029779-A2 EGF-GENISTEIN CONJUGATES FOR THE TREATMENT OF CANCER REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1997-08-21 WO disclosed
EP-0133225-B1 PEPTIDE DERIVATIVES AND THEIR SALTS, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, PROCESS AND INTERMEDIATES FOR THEIR PRODUCTION F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1988-10-19 EP disclosed
EP-0133225-A2 Peptide derivatives and their salts, pharmaceutical preparations containing them, process and intermediates for their production F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1985-02-20 EP disclosed
US-4410461-A Production of benzylic esters ASHLAND OIL, INC. (US) 1983-10-18 US disclosed
US-3862225-A D-RING SUBSTITUTED TETRACYCLINES PFIZER 1975-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250326731-A1 CATALYST-CONTROLLED SITE-SELECTIVE METHYLENE C-H LACTONIZATION OF DICARBOXYLIC ACIDS DNPH1, NISCH, PTMA CPA3 394/4885FOLH1 150/4885CYP1A2 3500/4885
US-20220348914-A1 OLIGONUCLEOTIDE-LIGAND CONJUGATES AND PROCESS FOR THEIR PREPARATION IGF2R, IRS1, INSR CPA3 4028/4885FOLH1 412/4885CYP1A2 4624/4885
US-12173288-B2 Oligonucleotide-ligand conjugates and process for their preparation IGF2R, IRS1, INSR CPA3 4028/4885FOLH1 412/4885CYP1A2 4624/4885
US-20250075208-A1 OLIGONUCLEOTIDE-LIGAND CONJUGATES AND PROCESS FOR THEIR PREPARATION IGF2R, IRS1, INSR CPA3 4028/4885FOLH1 412/4885CYP1A2 4624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.