SCHEMBL320738

SCHEMBL320738

O=S(=O)(Nc1ncc(F)cn1)c1cc(Cl)c(F)cc1F

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 4/20 0.56
SCN9A Q15858 7/20 0.48
SGK1 O00141 4/20 0.45
SCN3A Q9NY46 1/20 0.44
SCN1A P35498 3/20 0.40
SCN5A Q14524 3/20 0.40
SCN8A Q9UQD0 3/20 0.40
SCN1B Q07699 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20486322 0.87 SLC22A12 (0.48) SLC22A12SCN9ASGK1SCN3A
SCHEMBL20182483 0.72 SCN5A (0.62) SCN9ASCN1ASCN5ASCN8ASCN1B
SCHEMBL20238048 0.72 SCN8A (0.56) SCN9ASGK1SCN1ASCN5ASCN8A
SCHEMBL20238558 0.72 SCN5A (0.59) SLC22A12SCN9ASGK1SCN1ASCN5A
SCHEMBL19614071 0.72 SCN1A (0.65) SCN9ASCN1ASCN5ASCN8ASCN1B
SCHEMBL1095172 0.71 SCN5A (0.61) SCN9ASCN1ASCN5ASCN8ASCN1B
SCHEMBL30646286 0.71 ALPL (0.54) SCN9ASGK1
Hydrochloric Acid SCHEMBL20486310 0.71 SCN5A (0.60) SCN9ASCN1ASCN5ASCN8ASCN1B
SCHEMBL16757015 0.70 SCN1A (0.62) SCN9ASCN1ASCN5ASCN8A
SCHEMBL29668849 0.69 SCN9A (0.55) SLC22A12SCN9ASCN3ASCN1ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10316026-B2 Method for removing dimethoxybenzyl group DAIICHI SANKYO COMPANY, LIMITED (JP) 2019-06-11 US disclosed
US-9145407-B2 Sulfonamide compounds PFIZER LIMITED (GB) 2015-09-29 US disclosed
US-9145407-B2 Sulfonamide compounds PFIZER LIMITED (GB) 2015-09-29 US disclosed
US-9145407-B2 Sulfonamide compounds PFIZER LIMITED (GB) 2015-09-29 US disclosed
EP-2590972-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2015-01-21 EP disclosed
EP-2590972-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2015-01-21 EP disclosed
EP-2590972-A2 CHEMICAL COMPOUNDS Pfizer Limited (GB) 2013-05-15 EP disclosed
US-20130109667-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
US-20130109667-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
US-20130109667-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012004706-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-12 WO disclosed
WO-2012004706-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10316026-B2 Method for removing dimethoxybenzyl group DDT, ALKBH5, DDO SLC22A12 4678/4885SCN9A 3799/4885SGK1 2705/4885
US-20130109667-A1 Chemical Compounds SCN1A, SCN7A, SCN1B SLC22A12 1897/4885SCN9A 11/4885SGK1 995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.