SCHEMBL3244570

SCHEMBL3244570

CCc1cccc(C(=O)O)c1I

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLCN2 P51788 1/20 0.53
GABRA1 P14867 2/20 0.45
GABRB2 P47870 2/20 0.45
ALDH1A1 P00352 3/20 0.44
HMGB1 P09429 1/20 0.44
ALOX15 P16050 1/20 0.44
FOLH1 Q04609 2/20 0.44
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTT P42858 3/20 0.41
TSHR P16473 2/20 0.41
KAT6A Q92794 1/20 0.40
SLC16A3 O15427 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NR4A1 P22736 1/20 0.39
NR4A2 P43354 1/20 0.39
NR4A3 Q92570 1/20 0.39
MYC P01106 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27229008 0.84 ALDH1A1 (0.44) CLCN2ALDH1A1HMGB1ALOX15FOLH1
SCHEMBL21616779 0.83 BID (0.55) ALOX15KDM4EHSD17B10
SCHEMBL27571198 0.82 HMGB1 (0.51) CLCN2ALDH1A1HMGB1ALOX15FOLH1
SCHEMBL4368624 0.82 HMGB1 (0.43) CLCN2ALDH1A1HMGB1ALOX15FOLH1
SCHEMBL19834696 0.82 AKR1C3 (0.48) CLCN2ALDH1A1HPGDTDP1
Acetic Acid SCHEMBL29701125 0.81 GABRA1 (0.50) CLCN2GABRA1GABRB2ALOX15TDP1
SCHEMBL11322881 0.81 TSHR (0.59) ALDH1A1ALOX15FOLH1TSHR
SCHEMBL2443197 0.80 ALDH1A1 (0.60) ALDH1A1HMGB1ALOX15KDM4EHPGD
SCHEMBL4238088 0.80 KAT6A (0.54) CLCN2GABRA1GABRB2ALDH1A1HMGB1
SCHEMBL578127 0.79 CLCN2 (0.56) CLCN2GABRA1GABRB2ALDH1A1HMGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4284619-A INJECTING RADIOIODINE COMPOUND MEDI-PHYSICS, INC. (US) 1981-08-18 US claimed
CN-111433577-A Temperature detection label and article management device using same 株式会社日立制作所 2020-07-17 CN disclosed
US-9638690-B2 Compounds and compositions for use as alkylating agent sensors and methods of use thereof THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2017-05-02 US disclosed
US-20160131641-A1 COMPOUNDS AND COMPOSITIONS FOR USE AS ALKYLATING AGENT SENSORS AND METHODS OF USE THEREOF THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2016-05-12 US disclosed
EP-1799627-B1 IRON OR COBALT-CATALYZED CARBON-CARBON COUPLING REACTION OF ARYLS, ALKENES AND ALKINES WITH COPPER REAGENTS SALTIGO GMBH (DE) 2010-05-05 EP disclosed
US-7468378-B2 Substituted quinoline compounds PFIZER INC. (US) 2008-12-23 US disclosed
US-7393958-B2 Triamide-substituted heterobicyclic compounds PFIZER, INC. (US) 2008-07-01 US disclosed
US-7368573-B2 Triamide-substituted heterobicyclic compounds PFIZER INC. (US) 2008-05-06 US disclosed
EP-1799627-A1 IRON OR COBALT-CATALYZED CARBON-CARBON COUPLING REACTION OF ARYLS, ALKENES AND ALKINES WITH COPPER REAGENTS Ludwig-Maximilians-Universität München (DE) 2007-06-27 EP disclosed
US-20070093525-A1 Triamide-substituted heterobicyclic compounds PFIZER INC 2007-04-26 US disclosed
EP-0977734-A2 ARYLSECOCHOLADIENE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-02-09 EP disclosed
WO-1998047866-A2 ARYLSECOCHOLADIENE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1998-10-29 WO disclosed
WO-1995003700-A1 BRIDGED BIPHENYL CARBAPENEM ANTIBACTERIAL COMPOUNDS MERCK & CO., INC. (US) 1995-02-09 WO disclosed
WO-1995003699-A1 BRIDGED BIPHENYL CARBAPENEM COMPOUNDS AND METHODS OF USE MERCK & CO., INC. (US) 1995-02-09 WO disclosed
US-5374630-A Bridged carbapenem antibacterial compounds MERCK & CO., INC. (US) 1994-12-20 US disclosed
US-5372993-A Bridged carbapenem compounds, compositions containing such compounds and methods of use MERCK & CO., INC. (US) 1994-12-13 US disclosed
EP-0181526-B1 BENZOIC ACID DERIVATIVES Chugai Seiyaku Kabushiki Kaisha (JP) 1989-01-18 EP disclosed
US-4698364-A INFECTION CONTROL CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1987-10-06 US disclosed
EP-0181526-A1 Benzoic acid derivatives Chugai Seiyaku Kabushiki Kaisha (JP) 1986-05-21 EP disclosed
US-4020169-A FROM ARYL IODIDE OR BROMIDE AND TRIFLUOROMETHYL THIO COPPER MERCK & CO., INC. (US) 1977-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160131641-A1 COMPOUNDS AND COMPOSITIONS FOR USE AS ALKYLATING AGENT SENSORS AND METHODS OF USE THEREOF MGMT, MCL1, OGG1 CLCN2 1424/4885GABRA1 3516/4885GABRB2 4313/4885
US-20070093525-A1 Triamide-substituted heterobicyclic compounds APOB, MTPN, CTRB1 CLCN2 3889/4885GABRA1 2842/4885GABRB2 1237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.