SCHEMBL3244764

SCHEMBL3244764

Cc1ccc(CNC(=O)Cn2c(=O)n(C)c3cc(-c4cc(Cl)cc(Cl)c4)cnc32)o1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
GRIN1 Q05586 12/20 0.42
GRIN2B Q13224 12/20 0.42
ALDH1A1 P00352 4/20 0.40
HTT P42858 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 2/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13521574 0.84 TP53 (0.44) GRIN1GRIN2BMAPTMEN1KMT2A
SCHEMBL3114848 0.83 GRIN1 (0.43) GRIN1GRIN2BMAPT
SCHEMBL3129349 0.83 GRIN1 (0.48) CYP1A2CYP2D6CYP2C19GRIN1GRIN2B
SCHEMBL3118576 0.82 CES2 (0.49) GRIN1GRIN2BPOLBMAPT
SCHEMBL13521724 0.80 MAPT (0.49) GRIN1GRIN2BALDH1A1HTTSMN1; SMN2
SCHEMBL13521623 0.79 GRIN1 (0.49) GRIN1GRIN2BHTTHPGDPOLB
SCHEMBL13521710 0.79 GRIN1 (0.53) GRIN1GRIN2BPOLB
SCHEMBL3129279 0.79 KMT2A (0.50) ALDH1A1HTTSMN1; SMN2KDM4EPOLB
SCHEMBL3123200 0.79 ADORA2B (0.39) GRIN1GRIN2BHTTMAPT
SCHEMBL13521599 0.79 GRIN1 (0.44) GRIN1GRIN2BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO claimed