SCHEMBL3245236

SCHEMBL3245236

[O]c1ccc(-c2cscn2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.41
PARP1 P09874 1/20 0.40
KDM4A O75164 2/20 0.40
KDM4B O94953 2/20 0.40
KDM5C P41229 2/20 0.40
KDM5B Q9UGL1 2/20 0.40
ESR1 P03372 1/20 0.36
METAP1 P53582 3/20 0.36
TSHR P16473 2/20 0.36
METAP2 P50579 2/20 0.36
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.36
FKBP1A P62942 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6512842 0.80 RAB9A (0.47) CHEK2PARP1KDM4AKDM4BKDM5C
SCHEMBL496710 0.78 LTA4H (0.47) CHEK2PARP1KDM4AKDM4BKDM5C
SCHEMBL14754324 0.78 RAB9A (0.47) CHEK2PARP1METAP1METAP2KDM4E
SCHEMBL679357 0.78 METAP2 (0.46) METAP1METAP2KDM4ENPC1TP53
SCHEMBL18725070 0.78 TSHR (0.39) CHEK2PARP1KDM4AKDM4BKDM5C
SCHEMBL31126424 0.78 METAP2 (0.39) CHEK2PARP1KDM4AKDM4BKDM5C
SCHEMBL10284703 0.78 KMT2A (0.48) CHEK2PARP1METAP1TSHRMETAP2
SCHEMBL534208 0.78 ESR1 (0.42) CHEK2PARP1KDM4AKDM4BKDM5C
SCHEMBL679707 0.77 SCN9A (0.47) PARP1KDM4AKDM4BKDM5CKDM5B
SCHEMBL9231483 0.77 METAP1 (0.46) CHEK2PARP1KDM4AKDM4BKDM5C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1411935-B1 USE OF 4- (4-THIAZOLYL)PHENOXL ALKOXY-BENZAMIDINE DERIVATIVES FOR TREATMENT OF OSTEOPOROSIS DONG WHA PHARM CO LTD (KR) 2010-05-19 EP disclosed