SCHEMBL3245494

SCHEMBL3245494

CCCOC(=O)Oc1c[nH]c2c(=O)[nH]c3ccc(S(=O)(=O)NC4CCNCC4)cc3c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARG Q86W56 1/20 0.42
TDP1 Q9NUW8 3/20 0.39
BRAF P15056 1/20 0.38
TSHR P16473 1/20 0.36
KDR P35968 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 4/20 0.34
MAPT P10636 3/20 0.34
ALDH1A1 P00352 3/20 0.34
TP53 P04637 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
LMNA P02545 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GAA P10253 1/20 0.33
THRB P10828 1/20 0.33
CCR8 P51685 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ENPP2 Q13822 1/20 0.33
ATXN2 Q99700 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3253869 0.95 PARG (0.41) PARGTDP1BRAFTSHRKDR
SCHEMBL3251597 0.95 PARG (0.47) PARGTDP1BRAFTSHRCYP3A4
SCHEMBL3252200 0.95 PARG (0.41) PARGTDP1BRAFTSHRKDR
SCHEMBL3254875 0.94 PARG (0.43) PARGTDP1BRAFTSHRKDR
SCHEMBL3250757 0.90 PARG (0.46) PARGTDP1BRAFKDRPOLB
SCHEMBL3250591 0.88 PARG (0.48) PARGTDP1BRAFTSHRCYP3A4
SCHEMBL3250747 0.87 PARG (0.43) PARGTDP1BRAFTSHRKDR
SCHEMBL3250686 0.86 TDP1 (0.52) PARGTDP1TSHRCYP3A4CYP2C19
SCHEMBL3253874 0.86 TDP1 (0.52) PARGTDP1TSHRCYP3A4CYP2C19
SCHEMBL3245465 0.85 ALDH1A1 (0.36) POLBMAPTALDH1A1TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed