SCHEMBL3248358

SCHEMBL3248358

O=C(OC1(CCc2ccc(F)cc2)NC(c2cccc(F)c2)C(c2cccc(F)c2)N1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
CYP2C19 P33261 1/20 0.37
P2RX7 Q99572 2/20 0.34
CCR5 P51681 1/20 0.33
PKM P14618 1/20 0.33
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 1/20 0.32
CACNA1B Q00975 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PAX8 Q06710 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3253025 0.93 PAX8 (0.39) ALDH1A1CYP2C19CCR5PKMATM
SCHEMBL3257729 0.93 ALDH1A1 (0.40) ALDH1A1CYP2C19P2RX7PKMATM
SCHEMBL3256724 0.92 P2RX7 (0.39) ALDH1A1CYP2C19P2RX7PKMLMNA
SCHEMBL3253969 0.92 CYP2C19 (0.41) ALDH1A1CYP2C19L3MBTL1PAX8
SCHEMBL3258744 0.90 P2RX7 (0.38) ALDH1A1P2RX7LMNA
SCHEMBL3259173 0.90 ALDH1A1 (0.39) ALDH1A1CYP2C19P2RX7PKMATM
SCHEMBL3251176 0.89 ALDH1A1 (0.35) ALDH1A1CYP2C19P2RX7LMNAPAX8
SCHEMBL3252989 0.89 MTOR (0.40) ALDH1A1CYP2C19PKMPAX8
SCHEMBL3256527 0.88 ATM (0.45) ALDH1A1CYP2C19PKMATML3MBTL1
SCHEMBL3250310 0.88 P2RX7 (0.40) ALDH1A1CYP2C19P2RX7PKMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed