SCHEMBL3250310

SCHEMBL3250310

Cc1cccc(CCC2(OC(=O)C(F)(F)F)NC(c3cccc(F)c3)C(c3cccc(F)c3)N2)c1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.40
ALDH1A1 P00352 3/20 0.39
CYP2C19 P33261 1/20 0.37
PKM P14618 1/20 0.37
LMNA P02545 1/20 0.36
CACNA1B Q00975 1/20 0.36
DRD4 P21917 1/20 0.35
OPRM1 P35372 1/20 0.34
ALOX5 P09917 1/20 0.34
NR3C1 P04150 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3256724 0.93 P2RX7 (0.39) P2RX7ALDH1A1CYP2C19PKMLMNA
SCHEMBL3257729 0.91 ALDH1A1 (0.40) P2RX7ALDH1A1CYP2C19PKMLMNA
SCHEMBL3258350 0.91 SLC6A2 (0.39) CACNA1BALOX5
SCHEMBL3259233 0.88 P2RX7 (0.41) P2RX7ALDH1A1PKMLMNA
SCHEMBL3248358 0.88 ALDH1A1 (0.38) P2RX7ALDH1A1CYP2C19PKMLMNA
SCHEMBL3256527 0.86 ATM (0.45) ALDH1A1CYP2C19PKMLMNA
SCHEMBL3253969 0.86 CYP2C19 (0.41) ALDH1A1CYP2C19
SCHEMBL3251176 0.85 ALDH1A1 (0.35) P2RX7ALDH1A1CYP2C19LMNA
SCHEMBL3253025 0.85 PAX8 (0.39) ALDH1A1CYP2C19PKMOPRM1
SCHEMBL3252989 0.85 MTOR (0.40) ALDH1A1CYP2C19PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed