SCHEMBL3248495

SCHEMBL3248495

CCN(C(=O)C=Cc1ccc2[nH]c(=O)c3[nH]cc(C(=O)O)c3c2c1)C(=O)OC

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.35
ACHE P22303 4/20 0.35
MAOA P21397 3/20 0.35
MAOB P27338 3/20 0.35
GRIK1 P39086 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
GRIK2 Q13002 1/20 0.33
GRIK3 Q13003 1/20 0.33
KDM4E B2RXH2 4/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
POLB P06746 2/20 0.33
LMNA P02545 2/20 0.32
CYP1A2 P05177 2/20 0.32
MAPT P10636 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3253948 0.91 GABRA1 (0.37) BCHEACHEMAOAMAOBKDM4E
SCHEMBL3248903 0.81 TTR (0.45) MAOBGRIK1GRIA1GRIA2GRIA3
SCHEMBL3246027 0.81 TTR (0.45) MAOBGRIK1GRIA1GRIA2GRIA3
SCHEMBL3248489 0.79 MEN1 (0.41) MAOBKDM4EALDH1A1LMNACYP1A2
SCHEMBL3248486 0.79 MEN1 (0.41) MAOBKDM4EALDH1A1LMNACYP1A2
SCHEMBL3251013 0.76 GRIK1 (0.50) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL3251008 0.76 GRIK1 (0.50) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL3250563 0.75 MMP1 (0.49) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL3250568 0.75 MMP1 (0.49) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL3250273 0.74 TTR (0.45) MAOBKDM4EALDH1A1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP disclosed