SCHEMBL3248520

SCHEMBL3248520

O=C(O)CN1C(=O)CCc2cc(Br)cnc21

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ALDH1A1 P00352 4/20 0.37
ALOX12 P18054 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.35
GAA P10253 2/20 0.35
AKR1B1 P15121 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 2/20 0.34
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
CLK1 P49759 1/20 0.34
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25318355 0.82 HDAC1 (0.36) HDAC1HDAC8HDAC6ALDH1A1ALOX12
SCHEMBL30507436 0.82 HDAC1 (0.36) HDAC1HDAC8HDAC6ALDH1A1ALOX12
SCHEMBL3245592 0.81 ALDH1A1 (0.37) HDAC1HDAC8HDAC6ALDH1A1GAA
SCHEMBL30506707 0.78 HDAC1 (0.34) HDAC1HDAC8HDAC6ALDH1A1ALOX12
SCHEMBL25316939 0.78 HDAC1 (0.34) HDAC1HDAC8HDAC6ALDH1A1ALOX12
SCHEMBL3241068 0.78 CYP11B2 (0.41)
SCHEMBL3123128 0.77 HTT (0.49) ALDH1A1GAAAKR1B1TSHRMEN1
SCHEMBL26040102 0.76 BACE1 (0.35) HDAC1HDAC8HDAC6ALDH1A1MAPT
SCHEMBL4113410 0.74 HSD17B10 (0.38)
SCHEMBL3244879 0.74 LMNA (0.38) ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed