SCHEMBL3249374

SCHEMBL3249374

CCOC(=O)Oc1c[nH]c2c(=O)[nH]c3ccc(NC(C)=O)cc3c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.47
HPGD P15428 7/20 0.46
KDM4E B2RXH2 6/20 0.46
ALDH1A1 P00352 6/20 0.46
ESR1 P03372 1/20 0.46
MMP13 P45452 1/20 0.45
ADORA3 P0DMS8 1/20 0.43
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
HSD17B10 Q99714 3/20 0.43
KMT2A Q03164 2/20 0.43
ALOX15 P16050 1/20 0.43
ERCC1 P07992 1/20 0.42
DNASE1 P24855 1/20 0.42
FEN1 P39748 1/20 0.42
ERCC4 Q92889 1/20 0.42
PRNP P04156 1/20 0.41
LMNA P02545 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3243057 0.91 CHEK1 (0.37) CHEK1HPGDKDM4EALDH1A1ESR1
SCHEMBL3252205 0.90 TTK (0.42) CHEK1HPGDKDM4EALDH1A1ESR1
SCHEMBL3245415 0.90 CHEK1 (0.39) CHEK1HPGDKDM4EALDH1A1ESR1
SCHEMBL3241975 0.89 MEN1 (0.49) HPGDALDH1A1HSD17B10KMT2AALOX15
SCHEMBL3249852 0.89 BRD4 (0.52) KMT2AMAOASMN1; SMN2MEN1TP53
SCHEMBL3252529 0.89 ALDH1A1 (0.47) HPGDKDM4EALDH1A1HSD17B10KMT2A
SCHEMBL3256086 0.87 KDR (0.38) CHEK1HPGDKDM4EALDH1A1ESR1
SCHEMBL3254540 0.87 MMP2 (0.46) CHEK1HPGDKDM4EALDH1A1MMP13
SCHEMBL13928204 0.84 MMP13 (0.51) CHEK1HPGDKDM4EALDH1A1ESR1
SCHEMBL3245727 0.84 GABRA1 (0.50) HPGDALDH1A1HSD17B10KMT2APRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed