SCHEMBL3259233

SCHEMBL3259233

O=C(OC1(CCc2cccc(F)c2)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.41
PKM P14618 1/20 0.37
TAAR1 Q96RJ0 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
PPARG P37231 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM3 P20309 1/20 0.35
GPR52 Q9Y2T5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3256724 0.94 P2RX7 (0.39) P2RX7PKMTAAR1ALDH1A1LMNA
SCHEMBL3255000 0.90 P2RX7 (0.43) P2RX7PKMALDH1A1LMNAHCAR2
SCHEMBL3258350 0.88 SLC6A2 (0.39) CHRM2CHRM3GPR52
SCHEMBL3258394 0.88 P2RX7 (0.42) P2RX7TAAR1ALDH1A1HCAR2CHRM2
SCHEMBL3258744 0.88 P2RX7 (0.38) P2RX7ALDH1A1LMNA
SCHEMBL3250310 0.88 P2RX7 (0.40) P2RX7PKMALDH1A1LMNA
SCHEMBL3248358 0.87 ALDH1A1 (0.38) P2RX7PKMALDH1A1LMNA
SCHEMBL3251176 0.85 ALDH1A1 (0.35) P2RX7ALDH1A1LMNA
SCHEMBL3253025 0.84 PAX8 (0.39) PKMALDH1A1
SCHEMBL3257729 0.84 ALDH1A1 (0.40) P2RX7PKMALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed