SCHEMBL3255809

SCHEMBL3255809

Cc1cccc(CC2(OC(=O)C(F)(F)F)NC(c3ccccc3)C(c3ccccc3)N2)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
CACNA1B Q00975 1/20 0.36
SSTR4 P31391 1/20 0.35
ATM Q13315 1/20 0.35
RAB9A P51151 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CTBP2 P56545 1/20 0.34
CHRM2 P08172 2/20 0.34
CHRM3 P20309 2/20 0.34
GAA P10253 1/20 0.34
ORAI1 Q96D31 1/20 0.34
PKM P14618 1/20 0.34
TP53 P04637 1/20 0.34
CHRM1 P11229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3258350 0.90 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3CACNA1BATM
SCHEMBL3255000 0.87 P2RX7 (0.43) PKMTP53
SCHEMBL3253146 0.87 SMN1; SMN2 (0.37) ATMRAB9AMEN1KMT2AGAA
SCHEMBL3253979 0.84 CHRM5 (0.36) RAB9ACHRM2CHRM3GAATP53
SCHEMBL3253367 0.83 KDM1A (0.35) RAB9ACHRM3GAATP53CHRM1
SCHEMBL3256042 0.81 P2RX7 (0.39) ATMRAB9ACTBP2GAA
SCHEMBL3254057 0.81 TP53 (0.42) SLC6A2SLC6A4SLC6A3ATMRAB9A
SCHEMBL3250310 0.81 P2RX7 (0.40) CACNA1BPKM
SCHEMBL3258687 0.80 GPBAR1 (0.39) ATMKMT2AGAA
SCHEMBL3256725 0.80 GAA (0.33) RAB9AGAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed