SCHEMBL3253367

SCHEMBL3253367

O=C(OC1(Cc2ccc(F)c(F)c2)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.35
SIGMAR1 Q99720 2/20 0.35
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
ALDH1A1 P00352 3/20 0.33
TSHR P16473 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 2/20 0.32
HTT P42858 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GRM2 Q14416 1/20 0.31
GRM3 Q14832 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3257493 0.90 ALDH1A1 (0.38) ALDH1A1L3MBTL1
SCHEMBL3256757 0.90 RPA1 (0.34) GAARAB9AGRM2GRM3
SCHEMBL3253979 0.90 CHRM5 (0.36) CHRM5CHRM1CHRM3TP53GAA
SCHEMBL3254057 0.87 TP53 (0.42) KDM1AL3MBTL1TP53GAARAB9A
SCHEMBL3255000 0.86 P2RX7 (0.43) SIGMAR1ALDH1A1TP53
SCHEMBL3255018 0.86 GAA (0.35) ALDH1A1TP53GAARAB9ASMN1; SMN2
SCHEMBL3255278 0.84 SIGMAR1 (0.35) KDM1ASIGMAR1TP53GAAHTT
SCHEMBL3256725 0.83 GAA (0.33) KDM1ASIGMAR1TP53GAARAB9A
SCHEMBL3253146 0.83 SMN1; SMN2 (0.37) ALDH1A1L3MBTL1TP53GAARAB9A
SCHEMBL3258687 0.83 GPBAR1 (0.39) KDM1ASIGMAR1TSHRGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed