SCHEMBL3256385

SCHEMBL3256385

O=c1c(CN2CCNCC2)coc2cc(O)ccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.51
SIGMAR1 Q99720 2/20 0.49
ALDH1A1 P00352 9/20 0.46
TSHR P16473 2/20 0.46
RAB9A P51151 4/20 0.46
HSD17B10 Q99714 4/20 0.46
KDM4E B2RXH2 4/20 0.46
NPC1 O15118 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
HPGD P15428 3/20 0.46
MAOA P21397 2/20 0.46
CA12 O43570 1/20 0.46
AKR1B10 O60218 1/20 0.46
LMNA P02545 1/20 0.46
TTR P02766 1/20 0.46
ESR1 P03372 1/20 0.46
TP53 P04637 1/20 0.46
ALDH2 P05091 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251466 0.87 MAOA (0.51) XDHSIGMAR1ALDH1A1TSHRRAB9A
SCHEMBL3252425 0.86 SIGMAR1 (0.50) SIGMAR1ALDH1A1TSHRRAB9AHSD17B10
SCHEMBL3246823 0.83 SIGMAR1 (0.73) SIGMAR1ALDH1A1TSHRRAB9AHSD17B10
SCHEMBL3255205 0.82 ALDH1A1 (0.49) SIGMAR1ALDH1A1TSHRRAB9AHSD17B10
SCHEMBL13304409 0.81 ALDH1A1 (0.48) SIGMAR1ALDH1A1TSHRRAB9AHSD17B10
SCHEMBL3252433 0.77 ALDH1A1 (0.57) SIGMAR1ALDH1A1TSHRRAB9AHSD17B10
SCHEMBL3253325 0.76 ALDH1A1 (0.56) SIGMAR1ALDH1A1TSHRRAB9AHSD17B10
SCHEMBL21591575 0.75 MAOB (0.65) XDHALDH1A1RAB9AHSD17B10KDM4E
SCHEMBL3252274 0.75 ALDH1A1 (0.76) SIGMAR1ALDH1A1TSHRRAB9AHSD17B10
SCHEMBL3257338 0.73 ALDH1A1 (0.77) SIGMAR1ALDH1A1TSHRRAB9AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1890672-B1 USE OF CHROMONE DERIVATIVES MERCK PATENT GMBH (DE) 2010-06-02 EP disclosed
EP-1890672-B1 USE OF CHROMONE DERIVATIVES MERCK PATENT GMBH (DE) 2010-06-02 EP disclosed
EP-1890672-A1 USE OF CHROMONE DERIVATIVES Merck Patent GmbH (DE) 2008-02-27 EP disclosed
WO-2006128562-A1 USE OF CHROMONE DERIVATIVES MERCK PATENT GMBH (DE) 2006-12-07 WO disclosed