SCHEMBL3252425

SCHEMBL3252425

O=c1c(CN2CCOCC2)coc2cc(O)ccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.50
ALDH1A1 P00352 7/20 0.47
TSHR P16473 2/20 0.47
POLB P06746 2/20 0.47
GAA P10253 1/20 0.47
HSD17B10 Q99714 3/20 0.47
RAB9A P51151 3/20 0.47
CYP2C9 P11712 2/20 0.47
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
CA12 O43570 1/20 0.47
AKR1B10 O60218 1/20 0.47
LMNA P02545 1/20 0.47
TTR P02766 1/20 0.47
ESR1 P03372 1/20 0.47
TP53 P04637 1/20 0.47
ALDH2 P05091 1/20 0.47
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3253325 0.90 ALDH1A1 (0.56) SIGMAR1ALDH1A1TSHRPOLBGAA
SCHEMBL3251466 0.88 MAOA (0.51) SIGMAR1ALDH1A1TSHRPOLBHSD17B10
SCHEMBL3256385 0.86 XDH (0.51) SIGMAR1ALDH1A1TSHRPOLBGAA
SCHEMBL3246823 0.84 SIGMAR1 (0.73) SIGMAR1ALDH1A1TSHRPOLBHSD17B10
SCHEMBL3255205 0.83 ALDH1A1 (0.49) SIGMAR1ALDH1A1TSHRHSD17B10RAB9A
SCHEMBL13304409 0.82 ALDH1A1 (0.48) SIGMAR1ALDH1A1TSHRPOLBHSD17B10
SCHEMBL13072391 0.81 LTA4H (0.42) SIGMAR1ALDH1A1POLBHSD17B10CYP2C9
Oxazorone SCHEMBL29913823 0.78 TDP1 (0.66) ALDH1A1POLBGAAHSD17B10KDM4E
Oxazorone SCHEMBL2109280 0.78 TDP1 (0.66) ALDH1A1POLBGAAHSD17B10KDM4E
SCHEMBL3252433 0.78 ALDH1A1 (0.57) SIGMAR1ALDH1A1TSHRHSD17B10RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1890672-B1 USE OF CHROMONE DERIVATIVES MERCK PATENT GMBH (DE) 2010-06-02 EP disclosed
EP-1890672-A1 USE OF CHROMONE DERIVATIVES Merck Patent GmbH (DE) 2008-02-27 EP disclosed
WO-2006128562-A1 USE OF CHROMONE DERIVATIVES MERCK PATENT GMBH (DE) 2006-12-07 WO disclosed