SCHEMBL3255205

SCHEMBL3255205

CC(=O)N1CCN(Cc2coc3cc(O)ccc3c2=O)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.49
TSHR P16473 2/20 0.49
SIGMAR1 Q99720 2/20 0.49
P4HB P07237 1/20 0.48
RAB9A P51151 2/20 0.47
HSD17B10 Q99714 3/20 0.45
HTR1A P08908 1/20 0.44
LTA4H P09960 1/20 0.43
KDM4E B2RXH2 3/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43
CA12 O43570 1/20 0.43
AKR1B10 O60218 1/20 0.43
LMNA P02545 1/20 0.43
TTR P02766 1/20 0.43
ESR1 P03372 1/20 0.43
TP53 P04637 1/20 0.43
ALDH2 P05091 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3255333 0.91 ALDH1A1 (0.58) ALDH1A1TSHRSIGMAR1P4HBRAB9A
SCHEMBL13304409 0.90 ALDH1A1 (0.48) ALDH1A1TSHRSIGMAR1P4HBRAB9A
SCHEMBL3251466 0.84 MAOA (0.51) ALDH1A1TSHRSIGMAR1RAB9AHSD17B10
SCHEMBL3252425 0.83 SIGMAR1 (0.50) ALDH1A1TSHRSIGMAR1RAB9AHSD17B10
SCHEMBL3246823 0.82 SIGMAR1 (0.73) ALDH1A1TSHRSIGMAR1P4HBRAB9A
SCHEMBL3256385 0.82 XDH (0.51) ALDH1A1TSHRSIGMAR1RAB9AHSD17B10
SCHEMBL13856761 0.81 ALDH1A1 (0.74) ALDH1A1TSHRSIGMAR1RAB9AHSD17B10
SCHEMBL13304673 0.81 ALDH1A1 (0.57) ALDH1A1TSHRSIGMAR1P4HBRAB9A
SCHEMBL3252274 0.77 ALDH1A1 (0.76) ALDH1A1TSHRSIGMAR1RAB9AHSD17B10
SCHEMBL16408356 0.75 LTA4H (0.49) ALDH1A1TSHRP4HBRAB9AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1890672-B1 USE OF CHROMONE DERIVATIVES MERCK PATENT GMBH (DE) 2010-06-02 EP disclosed
EP-1890672-B1 USE OF CHROMONE DERIVATIVES MERCK PATENT GMBH (DE) 2010-06-02 EP disclosed
EP-1890672-A1 USE OF CHROMONE DERIVATIVES Merck Patent GmbH (DE) 2008-02-27 EP disclosed
WO-2006128562-A1 USE OF CHROMONE DERIVATIVES MERCK PATENT GMBH (DE) 2006-12-07 WO disclosed