SCHEMBL3258335

SCHEMBL3258335

O=C(OC1(Cc2ccc(F)cc2F)NC(c2cccc(F)c2)C(c2cccc(F)c2)N1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
CYP2C19 P33261 2/20 0.37
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
LMNA P02545 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
TRPA1 O75762 1/20 0.32
CACNA1B Q00975 1/20 0.32
TDP1 Q9NUW8 2/20 0.32
PKM P14618 1/20 0.32
P2RX7 Q99572 2/20 0.32
RECQL P46063 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3254884 0.92 SIGMAR1 (0.35) ALDH1A1HTR2AHTR2CTRPA1TDP1
SCHEMBL3255413 0.91 ALDH1A1 (0.38) ALDH1A1CYP2C19LMNACYP3A4MAPT
SCHEMBL3259173 0.88 ALDH1A1 (0.39) ALDH1A1CYP2C19LMNACYP3A4MAPT
SCHEMBL3257493 0.85 ALDH1A1 (0.38) ALDH1A1CYP2C19LMNACYP3A4MAPT
SCHEMBL3255278 0.83 SIGMAR1 (0.35) MAPTP2RX7
SCHEMBL3255755 0.82 ALDH1A1 (0.36) ALDH1A1CYP2C19CYP3A4MAPTCYP2C9
SCHEMBL3249024 0.82 KMT2A (0.41) ALDH1A1CYP2C19LMNAP2RX7
SCHEMBL3255000 0.81 P2RX7 (0.43) ALDH1A1LMNAPKMP2RX7
SCHEMBL3251110 0.81 ALDH1A1 (0.37) ALDH1A1CYP2C19LMNAMAPTCACNA1B
SCHEMBL3255401 0.81 P2RX7 (0.39) ALDH1A1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed