SCHEMBL3249024

SCHEMBL3249024

O=C(OC1(Cc2cccc(Cl)c2)NC(c2cccc(F)c2)C(c2cccc(F)c2)N1)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.41
MEN1 O00255 2/20 0.40
IDE P14735 1/20 0.40
P2RX7 Q99572 2/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.36
GRIN2B Q13224 1/20 0.35
HSD11B1 P28845 1/20 0.35
EPHX2 P34913 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRL1 P41146 1/20 0.35
NR3C1 P04150 1/20 0.35
HCRTR1 O43613 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3253134 0.90 HSD11B1 (0.39) KMT2AMEN1IDEP2RX7ALDH1A1
SCHEMBL3257493 0.88 ALDH1A1 (0.38) P2RX7ALDH1A1CYP2C19LMNA
SCHEMBL3255000 0.87 P2RX7 (0.43) P2RX7ALDH1A1LMNA
SCHEMBL3259173 0.87 ALDH1A1 (0.39) P2RX7ALDH1A1CYP2C19LMNA
SCHEMBL3256724 0.83 P2RX7 (0.39) P2RX7ALDH1A1CYP2C19LMNA
SCHEMBL3258335 0.82 ALDH1A1 (0.38) P2RX7ALDH1A1CYP2C19LMNA
SCHEMBL3255413 0.82 ALDH1A1 (0.38) P2RX7ALDH1A1CYP2C19LMNA
SCHEMBL3251176 0.82 ALDH1A1 (0.35) P2RX7ALDH1A1CYP2C19LMNA
SCHEMBL3258394 0.81 P2RX7 (0.42) KMT2AMEN1P2RX7ALDH1A1
SCHEMBL3256757 0.80 RPA1 (0.34) GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed