SCHEMBL3258394

SCHEMBL3258394

O=C(OC1(CCc2cccc(Cl)c2)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.42
ALDH1A1 P00352 3/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TRPV1 Q8NER1 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
ATM Q13315 1/20 0.36
PAX8 Q06710 1/20 0.36
PLAAT3 P53816 2/20 0.36
PLAAT5 Q96KN8 2/20 0.36
PLAAT2 Q9NWW9 2/20 0.36
PLAAT4 Q9UL19 2/20 0.36
GRM2 Q14416 1/20 0.36
GRM3 Q14832 1/20 0.36
POLB P06746 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
CHRM2 P08172 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3253134 0.90 HSD11B1 (0.39) P2RX7ALDH1A1KMT2AMEN1HPGD
SCHEMBL3259233 0.88 P2RX7 (0.41) P2RX7ALDH1A1TAAR1HCAR2CHRM2
SCHEMBL3255825 0.88 PDPK1 (0.36) ALDH1A1KMT2AMEN1TAAR1POLB
SCHEMBL3258561 0.87 PDPK1 (0.39) KMT2AMEN1TRPV1ATMPLAAT3
SCHEMBL3258350 0.87 SLC6A2 (0.39) KMT2AMEN1ATMGRM2GRM3
SCHEMBL3256724 0.83 P2RX7 (0.39) P2RX7ALDH1A1TAAR1HCAR2
SCHEMBL3258744 0.82 P2RX7 (0.38) P2RX7ALDH1A1KMT2AMEN1PLAAT3
SCHEMBL3253810 0.82 ALDH1A1 (0.41) ALDH1A1KMT2AMEN1SMN1; SMN2PLAAT3
SCHEMBL3253833 0.82 CES1 (0.41) P2RX7SMN1; SMN2POLBL3MBTL1
SCHEMBL3258306 0.81 P2RX7 (0.39) P2RX7ALDH1A1HPGDTRPV1PLAAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed