SCHEMBL3266768

SCHEMBL3266768

OC(CCCCCCc1ccccc1)n1cc(-c2ccco2)nn1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.43
FAAH O00519 1/20 0.43
DAGLA Q9Y4D2 1/20 0.40
SIRT1 Q96EB6 1/20 0.39
CACNA1B Q00975 1/20 0.38
APBA1 Q02410 1/20 0.38
ALDH1A1 P00352 2/20 0.38
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2161738 0.75 ALDH1A1 (0.47) CES1FAAHDAGLAALDH1A1NPC1
SCHEMBL2161819 0.70 CES1 (0.45) CES1FAAHDAGLA
SCHEMBL28331494 0.68 CYP19A1 (0.62) ALDH1A1NPC1TP53POLBRAB9A
SCHEMBL2161996 0.68 FAAH (0.47) CES1FAAH
SCHEMBL2162914 0.68 DAGLA (0.49) CES1FAAHDAGLAALDH1A1NPC1
SCHEMBL2162827 0.67 FAAH (0.40) CES1FAAH
SCHEMBL2161989 0.65 CES1 (0.61) CES1FAAHDAGLAALDH1A1
SCHEMBL16038331 0.63 ALDH1A1 (0.51) ALDH1A1NPC1POLBRAB9A
SCHEMBL4775723 0.63 TRPA1 (0.57) FAAH
SCHEMBL6471773 0.63 TRPA1 (0.57) FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010005572-A2 ALPHA-KETO HETEROCYCLES AS FAAH INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2010-01-14 WO disclosed