SCHEMBL3267545

SCHEMBL3267545

CN1CCC(C(=O)N2CCN(Cc3cccc4cc(C(=O)O)n(C)c34)CC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
RORC P51449 2/20 0.43
DHODH Q02127 2/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
TSHR P16473 3/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ADRB2 P07550 1/20 0.42
MTNR1B P49286 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27856261 0.96 MEN1 (0.44) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL690572 0.91 RORC (0.40) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL27856266 0.88 KMT2A (0.46) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL3233896 0.88 RORC (0.40) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL3267550 0.86 MTNR1B (0.43) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL3267160 0.86 FAAH (0.38) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL690228 0.84 EPHX2 (0.42) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL3228834 0.84 EPHX2 (0.42) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL689275 0.84 EPHX2 (0.42) ALDH1A1RORCDHODHMEN1KMT2A
SCHEMBL27856260 0.83 HTR1A (0.42) ALDH1A1MEN1KMT2AALOX15SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102186818-B 7-(piperazine-1-ymethyl)-1h-indole-2-carboxylic acid (phenyl)-amide derivatives and allied compounds as p38 map kinase inhibitors for the treatment of respiratory diseases BOEHRINGER INGELHEIM INT 2013-10-02 CN disclosed
CN-102186818-A 7-(piperazine-1-ymethyl)-1h-indole-2-carboxylic acid (phenyl)-amide derivatives and allied compounds as p38 map kinase inhibitors for the treatment of respiratory diseases BOEHRINGER INGELHEIM INT 2011-09-14 CN disclosed
WO-2010026096-A1 7-(PIPERAZINE-1-YMETHYL)-1H-INDOLE-2-CARBOXYLIC ACID (PHENYL)-AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHIBITORS FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-03-11 WO disclosed