SCHEMBL3268660

SCHEMBL3268660

COC(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA1 P56199 3/20 0.68
MAPK1 P28482 1/20 0.58
CMA1 P23946 1/20 0.58
HDAC1 Q13547 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
LMNA P02545 2/20 0.56
HPGD P15428 2/20 0.56
MEN1 O00255 1/20 0.55
MAPT P10636 1/20 0.55
ALOX12 P18054 1/20 0.55
KMT2A Q03164 1/20 0.55
NLRP1 Q9C000 1/20 0.55
FLT1 P17948 1/20 0.55
FLT4 P35916 1/20 0.55
KDR P35968 1/20 0.55
ALPL P05186 2/20 0.54
TP53 P04637 1/20 0.53
PPARG P37231 2/20 0.53
IDH1 O75874 1/20 0.53
ACLY P53396 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4565254 0.87 IKBKB (0.67) ITGA1MAPK1HDAC1HDAC8LMNA
SCHEMBL13631960 0.81 ITGA1 (1.00) ITGA1MAPK1HDAC1HDAC8LMNA
SCHEMBL4815316 0.80 ITGA1 (0.67) ITGA1MAPK1HDAC1HDAC8LMNA
SCHEMBL14018772 0.80 MAPT (0.63) ITGA1MAPK1HDAC1HDAC8LMNA
SCHEMBL21545964 0.79 NR4A2 (0.55) ITGA1MAPK1CMA1LMNAHPGD
SCHEMBL8274502 0.79 HDAC1 (0.74) ITGA1MAPK1HDAC1HDAC8
SCHEMBL4882914 0.77 PGR (0.61) ITGA1MAPK1HDAC1HDAC8LMNA
SCHEMBL4880041 0.77 SGK1 (0.55) ITGA1HDAC1HDAC8LMNAMEN1
SCHEMBL94831 0.77 MAPT (0.63) ITGA1MAPK1HDAC1HDAC8LMNA
SCHEMBL28121241 0.77 MAPT (0.63) ITGA1MAPK1HDAC1HDAC8LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1914229-B1 NOVEL CERCOSPORAMIDE DERIVATIVE DAIICHI SANKYO CO LTD (JP) 2010-06-16 EP disclosed
US-20090036492-A1 Novel Cercosporamide Derivative DAIICHI SANKYO COMPANY, LIMITED (JP) 2009-02-05 US disclosed
EP-1914229-A1 NOVEL CERCOSPORAMIDE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2008-04-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036492-A1 Novel Cercosporamide Derivative GPR119, CBR3, SLC5A2 ITGA1 3624/4885MAPK1 167/4885CMA1 468/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.