SCHEMBL3269356

SCHEMBL3269356

NC(=O)Oc1[nH]c2sc(Sc3ccccc3)nc2c1Sc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 3/20 0.35
DHFR P00374 2/20 0.35
TUBB4A P04350 4/20 0.33
TUBB P07437 4/20 0.33
TUBA3C P0DPH7 4/20 0.33
TUBA1B P68363 4/20 0.33
TUBA4A P68366 4/20 0.33
TUBB4B P68371 4/20 0.33
TUBB3 Q13509 4/20 0.33
TUBB2A Q13885 4/20 0.33
TUBB8 Q3ZCM7 4/20 0.33
TUBA3E Q6PEY2 4/20 0.33
TUBA1A Q71U36 4/20 0.33
TUBA1C Q9BQE3 4/20 0.33
TUBB6 Q9BUF5 4/20 0.33
TUBB2B Q9BVA1 4/20 0.33
TUBB1 Q9H4B7 4/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3269846 0.87 TYMS (0.39) TYMSDHFRTUBB4ATUBBTUBA3C
SCHEMBL3272659 0.86 EDNRA (0.44) DHFRTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL3173374 0.81 TYMS (0.39) TYMSDHFRTUBB4ATUBBTUBA3C
SCHEMBL3274436 0.80 SIRT1 (0.35) TYMSDHFRTUBB4ATUBBTUBA3C
SCHEMBL3269941 0.75 TYMS (0.41) TYMSTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL3270007 0.75 EDNRA (0.44) DHFRTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL3269782 0.75 TYMS (0.41) TYMSDHFRTUBB4ATUBBTUBA3C
SCHEMBL3270312 0.74 TNKS2 (0.39) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL4035502 0.73 TUBB4A (0.39) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL3268800 0.72 RHEB (0.39) TYMSTUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784409-B1 SUBSTITUTED THIENOPYRROLE CARBOXYLIC ACID AMIDES, PYRROLOTHIAZOLE CARBOXYLIC ACID AMIDES, AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2010-06-16 EP claimed