Aminothiazole

Aminothiazole

SCHEMBL3269558

Nc1nccs1.O=S(=O)(O)O

nearest known ligand 0.71

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Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Aminothiazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A known ✓ P35348 1/20 0.41
ALDH1A1 P00352 4/20 0.71
TSHR P16473 1/20 0.71
NOS1 P29475 1/20 0.71
HSD17B10 Q99714 1/20 0.71
ACP1 P24666 3/20 0.43
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP2C9 P11712 1/20 0.41
EDNRA P25101 1/20 0.41
SLC6A4 P31645 1/20 0.41
PRMT6 Q96LA8 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP2C19 P33261 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
RECQL P46063 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
FBP1 P09467 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aminothiazole SCHEMBL27899272 0.85
Aminothiazole SCHEMBL7401 0.84
Aminothiazole SCHEMBL10428703 0.84
Aminothiazole SCHEMBL4962431 0.84 ALDH1A1 (1.00) ALDH1A1TSHRNOS1HSD17B10LMNA
Aminothiazole SCHEMBL1241596 0.83 ALDH1A1 (0.75) ALDH1A1TSHRNOS1HSD17B10ACP1
Aminothiazole SCHEMBL27943753 0.82
Aminothiazole SCHEMBL29012817 0.82
Aminothiazole SCHEMBL28159425 0.82
Aminothiazole SCHEMBL7473421 0.82
Aminothiazole SCHEMBL2350289 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-220048138-U Reaction device for continuously producing 2-bromothiazole 济南悟通生物科技有限公司 2023-11-21 CN disclosed
CN-109942600-A A kind of preparation method of Yi Dushaban 内蒙古京东药业有限公司 2019-06-28 CN disclosed
EP-1241232-B1 METAL CHELATE DYESTUFF FOR INK JET RECORDING AND WATER-BASE INK JET RECORDING FLUID CONTAINING THE SAME MITSUBISHI CHEM CORP (JP) 2010-06-16 EP disclosed
US-6755903-B2 FORMED FROM AN AZO COMPOUND CONTAINING AN N-HETEROARYL RING, E.G., IMIDAZOLE, AND AN OPTIONALLY SUBSTITUTED NAPHTHYL RING AND PREFERABLY A COPPER, NICKEL OR COBALT COMPOUND MITSUBISHI CHEMICAL CORPORATION (JP) 2004-06-29 US disclosed
US-20030088077-A1 Formed from an azo compound containing an N-heteroaryl ring, e.g., imidazole, and an optionally substituted naphthyl ring and preferably a copper, nickel or cobalt compound MITSUBISHI CHEMICAL CORPORATION (JP) 2003-05-08 US disclosed
EP-1241232-A1 METAL CHELATE DYESTUFF FOR INK JET RECORDING AND WATER-BASE INK JET RECORDING FLUID CONTAINING THE SAME MITSUBISHI CHEMICAL CORPORATION (JP) 2002-09-18 EP disclosed
EP-0314046-B1 Method of quantitative analysis of hydrogen peroxide and reagent therefor DAIICHI PURE CHEMICALS CO LTD (JP) 1994-06-01 EP disclosed
US-4933277-A Method of quantitative analysis of hydrogen peroxide and reagent therefor DAIICHI PURE CHEMICALS CO., LTD. (JP) 1990-06-12 US disclosed
EP-0314046-A2 Method of quantitative analysis of hydrogen peroxide and reagent therefor DAIICHI PURE CHEMICALS CO. LTD. (JP) 1989-05-03 EP disclosed
US-4046752-A Process for preparing an azo compound from a 2-aminothiazole diazo component HOECHST AKTIENGESELLSCHAFT (DT) 1977-09-06 US disclosed