SCHEMBL3274573

SCHEMBL3274573

Cc1ccc([CH]Cc2ccc(F)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 3/20 0.57
ACHE P22303 2/20 0.52
KMT2A Q03164 5/20 0.46
MEN1 O00255 3/20 0.46
BCHE P06276 1/20 0.45
TRPA1 O75762 1/20 0.43
CYP2A6 P11509 1/20 0.41
ALDH1A1 P00352 3/20 0.41
HTT P42858 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 3/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RAB9A P51151 1/20 0.40
GLA P06280 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5056468 0.89 CYP2A6 (0.50) NFE2L2ACHECYP2A6KDM4ESMN1; SMN2
SCHEMBL8364378 0.89 TRPA1 (0.45) NFE2L2KMT2ATRPA1RAB9A
SCHEMBL21179476 0.87 CYP2A6 (0.48) NFE2L2ACHECYP2A6KDM4ESMN1; SMN2
SCHEMBL16178490 0.80 MAPT (0.49) KMT2AMEN1TRPA1ALDH1A1HTT
SCHEMBL16225102 0.79 LMNA (0.44) KMT2AMEN1TRPA1HTTLMNA
SCHEMBL5360664 0.79 NFE2L2 (0.61) NFE2L2KMT2AMEN1CYP2A6ALDH1A1
SCHEMBL3241749 0.79 LMNA (0.42) ACHEBCHECYP2A6ALDH1A1HTT
SCHEMBL654153 0.79 NFE2L2 (0.52) NFE2L2ACHEKMT2AMEN1BCHE
SCHEMBL8210813 0.79 NFE2L2 (0.52) NFE2L2KMT2AMEN1TRPA1CYP2A6
SCHEMBL1987774 0.79 MAOB (0.46) ACHEBCHECYP2A6ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1278737-B1 PROCESS AND INTERMEDIATES FOR MAKING SUBSTITUTED ASPARTIC ACID ACETALS VERTEX PHARMA (US) 2010-06-30 EP claimed