SCHEMBL8364378

SCHEMBL8364378

Fc1ccc([CH]Cc2ccc(F)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.45
IDO1 P14902 5/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
TAAR1 Q96RJ0 3/20 0.41
NFE2L2 Q16236 2/20 0.41
KMT2A Q03164 1/20 0.41
AGXT P21549 2/20 0.39
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
HSD11B1 P28845 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3274573 0.89 NFE2L2 (0.57) TRPA1NFE2L2KMT2ARAB9A
SCHEMBL16178490 0.89 MAPT (0.49) TRPA1KMT2ANPC1RAB9A
SCHEMBL8210813 0.89 NFE2L2 (0.52) TRPA1IDO1LOXL2NFE2L2KMT2A
SCHEMBL654153 0.89 NFE2L2 (0.52) TRPA1NFE2L2KMT2AMAOB
SCHEMBL5557951 0.85 L3MBTL1 (0.41) TRPA1IDO1LOXL2KMT2ANPC1
SCHEMBL16225102 0.84 LMNA (0.44) TRPA1KMT2AHSD11B1NPC1RAB9A
SCHEMBL5360664 0.84 NFE2L2 (0.61) NFE2L2KMT2AMAOAMAOB
SCHEMBL14880614 0.81 TAAR1 (0.48) TRPA1IDO1LOXL2TAAR1NFE2L2
SCHEMBL5941183 0.79 NFE2L2 (0.50) IDO1TAAR1NFE2L2AGXTMAOA
SCHEMBL154188 0.79 NFE2L2 (0.55) LOXL2TAAR1NFE2L2MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106946974-B Ursolic amide derivative containing pyrazole heterocycle and synthesis and application thereof 中国科学院上海高等研究院 2020-03-31 CN disclosed
EP-0929217-A4 SORDARIN DERIVATIVES MERCK & CO INC (US) 1999-12-15 EP disclosed
EP-0929217-A1 SORDARIN DERIVATIVES Merck & Co., Inc. (US) 1999-07-21 EP disclosed
US-5811422-A USEFUL FOR TREATING VIRAL INFECTIONS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-09-22 US disclosed
WO-1998015178-A1 SORDARIN DERIVATIVES MERCK & CO., INC. (US) 1998-04-16 WO disclosed
US-5610294-A VIRAL TREATMENT THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-11 US disclosed