SCHEMBL3282871

SCHEMBL3282871

NC(=O)c1c(S(=O)(=O)N2CC3CN(CC[CH]c4ccccc4)CC3C2)cnn1-c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK2 O43353 1/20 0.36
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SLC9A1 P19634 2/20 0.32
SLC9A2 Q9UBY0 2/20 0.32
ACLY P53396 1/20 0.32
PTGS1 P23219 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
LOX P28300 1/20 0.32
PTGS2 P35354 1/20 0.32
CA9 Q16790 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
FPR1 P21462 1/20 0.31
HPGD P15428 1/20 0.31
MAPT P10636 1/20 0.31
HSD11B1 P28845 1/20 0.31
MAPK14 Q16539 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694243 1.00 RIPK2 (0.36) RIPK2NPC1RAB9ASLC9A1SLC9A2
SCHEMBL4690864 0.83 RIPK2 (0.40) RIPK2NPC1RAB9ASLC9A1SLC9A2
SCHEMBL4693316 0.78 EIF4A3 (0.39) RIPK2RAB9APTGS1CA12CA1
SCHEMBL4691488 0.75 FPR2 (0.37) HPGDMAPT
SCHEMBL4694244 0.72 EIF4A3 (0.45) SLC9A1SLC9A2PTGS2HPGDMAPT
SCHEMBL4695049 0.71 TSHR (0.39) HPGDMEN1KMT2A
SCHEMBL4691594 0.71 FPR2 (0.34) ACLYMAPT
SCHEMBL4691732 0.70 KDM4E (0.43) KEAP1NFE2L2MAPTHSD11B1MAPK14
SCHEMBL4694498 0.70 CCR5 (0.37)
SCHEMBL4692781 0.70 PKM (0.36) HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7714018-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2010-05-11 US disclosed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
US-7164019-B2 Such as cyclopentanecarboxylic acid {(S)-1-phenyl-3-[5-(pyridine-3-carbonyl)-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl]-propyl}-amide; antagonists of chemokine receptors, useful for treating/preventing human immunodeficiency virus infection, AIDS or ARC ROCHE PALO ALTO LLC (US) 2007-01-16 US disclosed
US-20060014767-A1 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC 2006-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060014767-A1 Heterocyclic antiviral compounds CCR5, ACKR3, CXCR1 RIPK2 212/4885NPC1 246/4885RAB9A 1690/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.