Talibegron

Talibegron

SCHEMBL328977

O=C(O)Cc1ccc(OCCNC[C@H](O)c2ccccc2)cc1

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.97
ADRB3 P13945 14/20 0.56
ADRB1 P08588 6/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
KDM4E B2RXH2 1/20 0.56
GAA P10253 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
CYP1A2 P05177 1/20 0.54
ADRB2 P07550 1/20 0.54
ALDH1A1 P00352 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Talibegron SCHEMBL3699503 1.00 ALOX15 (0.97) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
Talibegron SCHEMBL6060362 1.00 ALOX15 (0.97) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
Talibegron SCHEMBL1230810 0.99 ALOX15 (1.00) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
Talibegron SCHEMBL8976330 0.99 ALOX15 (1.00) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
SCHEMBL8976026 0.90 ALOX15 (0.80) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
SCHEMBL8976032 0.90 ALOX15 (0.80) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
SCHEMBL8976399 0.89 ALOX15 (0.78) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL8976317 0.89 ALOX15 (0.82) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL8976435 0.89 ALOX15 (0.82) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E
SCHEMBL8976401 0.89 ALOX15 (0.78) ALOX15ADRB3ADRB1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 586 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230158028-A1 COMPOUNDS AND METHODS FOR INDUCING UCP1 EXPRESSION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-05-25 US claimed
EP-4132914-A1 COMPOUNDS AND METHODS FOR INDUCING UCP1 EXPRESSION The Regents of the University of California (US) 2023-02-15 EP claimed
US-11136342-B2 Carbonate prodrugs and methods of using the same ACORDA THERAPEUTICS, INC. (US) 2021-10-05 US claimed
US-20200157126-A1 CARBONATE PRODRUGS AND METHODS OF USING THE SAME ACORDA THERAPEUTICS, INC. 2020-05-21 US claimed
US-10377779-B2 Carbonate prodrugs and methods of using the same ACORDA THERAPEUTICS, INC. (US) 2019-08-13 US claimed
US-20180086778-A1 CARBONATE PRODRUGS AND METHODS OF USING THE SAME NEUROGESX, INC. 2018-03-29 US claimed
EP-2961730-A2 METHOD OF MAKING 1-(ACYLOXY)-ALKYL CARBAMATE COMPOUNDS XenoPort, Inc. (US) 2016-01-06 EP claimed
US-20150158809-A9 METHOD OF MAKING 1-(ACYLOXY)-ALKYL CARBAMATE COMPOUNDS XENOPORT, INC. (US) 2015-06-11 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
CN-104427985-A Pharmaceutical combination for the treatment of metabolic disorders BOEHRINGER INGELHEIM INT 2015-03-18 CN claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
EP-2124970-A1 PHARMACEUTICAL COMPOSITION COMPRISING A PYRAZOLE-O-GLUCOSIDE DERIVATIVE Boehringer Ingelheim International GmbH (DE) 2009-12-02 EP claimed
WO-2009143297-A1 CARBONATE PRODRUGS AND METHODS OF USING THE SAME NEUROGESX, INC. (US) 2009-11-26 WO claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2008087198-A1 PHARMACEUTICAL COMPOSITION COMPRISING A PYRAZOLE-O-GLUCOSIDE DERIVATIVE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-24 WO claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-0516349-B1 2-Hydroxy-2-phenylethylamine derivatives as beta-3-adrenoceptor agonists ZENECA LTD (GB) 1995-09-20 EP claimed
US-5393779-A Anti-obesity, hypoglycemic, adrenergic blocking agents ZENECA LIMITED (GB) 1995-02-28 US claimed
EP-0516349-A2 2-Hydroxy-2-phenylethylamine derivatives as beta-3-adrenoceptor agonists ZENECA LIMITED (GB) 1992-12-02 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230158028-A1 COMPOUNDS AND METHODS FOR INDUCING UCP1 EXPRESSION TFAM, FABP4, CPT2 ALOX15 627/4885ADRB3 83/4885ADRB1 106/4885
US-20200157126-A1 CARBONATE PRODRUGS AND METHODS OF USING THE SAME CA6, CA7, CA4 ALOX15 1963/4885ADRB3 4025/4885ADRB1 4090/4885
US-20150158809-A9 METHOD OF MAKING 1-(ACYLOXY)-ALKYL CARBAMATE COMPOUNDS CPS1, CA7, NAAA ALOX15 1062/4885ADRB3 3450/4885ADRB1 3375/4885
US-11136342-B2 Carbonate prodrugs and methods of using the same CA6, CA7, CA4 ALOX15 1963/4885ADRB3 4025/4885ADRB1 4090/4885
US-10377779-B2 Carbonate prodrugs and methods of using the same CA6, CA7, CA4 ALOX15 1963/4885ADRB3 4025/4885ADRB1 4090/4885
US-20180086778-A1 CARBONATE PRODRUGS AND METHODS OF USING THE SAME CA6, CA7, CA4 ALOX15 1963/4885ADRB3 4025/4885ADRB1 4090/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.