SCHEMBL3302277

SCHEMBL3302277

CCCN(CCC)c1ccc(CC)c([N+](=O)[O-])c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.50
TSHR P16473 2/20 0.50
CYP3A4 P08684 2/20 0.50
MAPK1 P28482 2/20 0.50
ALDH3A1 P30838 2/20 0.48
HCAR3 P49019 3/20 0.47
ALDH1A1 P00352 3/20 0.46
PDK1 Q15118 1/20 0.46
VCAM1 P19320 3/20 0.40
MAPT P10636 4/20 0.40
CYP1A2 P05177 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
AR P10275 1/20 0.36
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3286485 0.84 TSHR (0.50) TDP1TSHRCYP3A4MAPK1ALDH3A1
SCHEMBL22897851 0.83 TDP1 (0.49) TDP1TSHRCYP3A4MAPK1ALDH3A1
SCHEMBL22115093 0.83 TSHR (0.51) TDP1TSHRCYP3A4MAPK1ALDH3A1
SCHEMBL29560800 0.83 TDP1 (0.49) TDP1TSHRCYP3A4MAPK1ALDH3A1
SCHEMBL3054634 0.81 MAPT (0.63) TDP1TSHRCYP3A4MAPK1ALDH3A1
SCHEMBL12848080 0.80 PDK1 (0.51) TDP1TSHRALDH3A1HCAR3ALDH1A1
SCHEMBL3053127 0.79 HCAR3 (0.49) TDP1TSHRCYP3A4MAPK1ALDH3A1
SCHEMBL3054662 0.79 VCAM1 (0.51) TDP1TSHRCYP3A4MAPK1ALDH3A1
SCHEMBL22897786 0.78 HCAR3 (0.45) TDP1TSHRCYP3A4MAPK1ALDH3A1
SCHEMBL27737624 0.77 ALDH1A1 (0.59) TDP1TSHRCYP3A4MAPK1HCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7714009-B2 Nitrogen-containing fused heterocyclic compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-11 US disclosed
US-20070135452-A1 Nitrogen-containing fused heterocyclic compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070135452-A1 Nitrogen-containing fused heterocyclic compounds NPY4R, NR4A3, NR3C2 TDP1 4581/4885TSHR 278/4885CYP3A4 428/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.